Compile Data Set for Download or QSAR
maximum 50k data
Found 158 Enz. Inhib. hit(s) with all data for entry = 9048
LigandPNGBDBM281483(US10022387, Example 8 | US10596184, Example 8 | US...)
Affinity DataIC50: >100nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281540(US10022387, Example 66 | US10596184, Example 66 | ...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281541(US10022387, Example 67 | US10596184, Example 67 | ...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281541(US10022387, Example 67 | US10596184, Example 67 | ...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281542(US10022387, Example 68 | US10596184, Example 68 | ...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281542(US10022387, Example 68 | US10596184, Example 68 | ...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM294399(2-(1H-Benzo[d]imidazol- 2-yl)-6-(6-fluoro- 5-metho...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM294402(2-(1H-Benzo[d]imidazol- 2-yl)-6-(5-(dimethyl- phos...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM294402(2-(1H-Benzo[d]imidazol- 2-yl)-6-(5-(dimethyl- phos...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281550(N-(5-(2-(1H-Benzo[d]imidazol-2- yl)benzo[d]oxazol-...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281550(N-(5-(2-(1H-Benzo[d]imidazol-2- yl)benzo[d]oxazol-...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281549(N-(5-(2-(1H-Benzo[d]imidazol-2- yl)benzo[d]oxazol-...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281549(N-(5-(2-(1H-Benzo[d]imidazol-2- yl)benzo[d]oxazol-...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281550(N-(5-(2-(1H-Benzo[d]imidazol-2- yl)benzo[d]oxazol-...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281550(N-(5-(2-(1H-Benzo[d]imidazol-2- yl)benzo[d]oxazol-...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281551(N-(5-(2-(1H-Benzo[d]imidazol-2- yl)benzo[d]oxazol-...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281553(N-(5-(2-(1H-Benzo[d]imidazol-2- yl)benzo[d]oxazol-...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281553(N-(5-(2-(1H-Benzo[d]imidazol-2- yl)benzo[d]oxazol-...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281554(US10022387, Example 80 | US10596184, Example 80 | ...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM294335(2-(1H-Benzo[d]imidazol-2-yl)-6-(5-methoxypyridin-3...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281479(US10022387, Example 4 | US10022387, Example 5 | US...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281485(US10022387, Example 11 | US10596184, Example 11 | ...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281486(US10022387, Example 12 | US10596184, Example 12 | ...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281488(US10022387, Example 14 | US10596184, Example 14 | ...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281490(US10022387, Example 16 | US10596184, Example 16 | ...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM437712(N-(5-(2-(1H- Benzo[d]imidazol- 2-yl)benzo[d]oxazol...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM437712(N-(5-(2-(1H- Benzo[d]imidazol- 2-yl)benzo[d]oxazol...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281492(N-(5-(2-(1H- Benzo[d]imidazol- 2- yl)benzo[d]oxazo...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281493(N-(5-(2-(1H- Benzo[d]imidazol- 2- yl)benzo[d]oxazo...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281493(N-(5-(2-(1H- Benzo[d]imidazol- 2- yl)benzo[d]oxazo...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM294350(N-(5-(2-(1H- Benzo[d]imidazol-2- yl)benzo[d]oxazol...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281495(N'-{5-[2-(1H- Benzimidazol-2- yl)-1,3- benzoxazol-...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281496(N'-{5-[2-(1H- Benzimidazol-2- yl)-1,3- benzoxazol-...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281496(N'-{5-[2-(1H- Benzimidazol-2- yl)-1,3- benzoxazol-...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281497(N'-{5-[2-(1H- Benzimidazol-2- yl)-1,3- benzoxazol-...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281497(N'-{5-[2-(1H- Benzimidazol-2- yl)-1,3- benzoxazol-...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281498(N-(5-(2-(1H- Benzo[d]imidazol- 2 - yl)benzo[d]oxaz...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281499(N-(5-(2-(1H- Benzo[d]imidazol- 2 - yl)benzo[d]oxaz...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281499(N-(5-(2-(1H- Benzo[d]imidazol- 2 - yl)benzo[d]oxaz...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281500(N-(5-(2-(1H- Benzo[d]imidazol- 2 - yl)benzo[d]oxaz...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281501(N-(5-(2-(1H- Benzo[d]imidazol- 2 - yl)benzo[d]oxaz...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281502(N-(5-(2-(1H- Benzo[d]imdiazol- 2 - yl)benzo[d]oxaz...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281502(N-(5-(2-(1H- Benzo[d]imdiazol- 2 - yl)benzo[d]oxaz...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281503(N-(5-(2-(1H- Benzo[d]imidazol- 2- yl)benzo[d]oxazo...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281503(N-(5-(2-(1H- Benzo[d]imidazol- 2- yl)benzo[d]oxazo...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281504(N-(5-(2-(1H- Benzo[d]imidazol- 2 - yl)benzo[d]oxaz...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281504(N-(5-(2-(1H- Benzo[d]imidazol- 2 - yl)benzo[d]oxaz...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM437727(2-(1H-Benzimidazol-2-yl)-6-(1-ethyl-1H-indazol-6-y...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM437727(2-(1H-Benzimidazol-2-yl)-6-(1-ethyl-1H-indazol-6-y...)
Affinity DataIC50: <250nMAssay Description:PI3Kdelta: The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM281506(N-(5-(2-(1H- Benzo[d]imidazol- 2- yl)benzo[d]oxazo...)
Affinity DataIC50: <250nMAssay Description:PI3K-gamma:The kinase reaction was conducted in polystyrene 384-well Greiner Bio-one white plate from Thermo Fisher Scientific in a final volume of 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 158 total ) | Next | Last >>
Jump to: