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Patent code US10781211

Compile Data Set for Download or QSAR

Found 677 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280477
PNG
(US10030020, Example 22 | US10781211, Example 22)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(cc3N3CCOCC3)C(F)(F)F)C2)CC1)C(F)(F)F
Show InChI InChI=1S/C24H28F9N3O3/c25-22(26,27)17-2-1-16(18(13-17)35-9-11-38-12-10-35)14-34-6-3-21(15-34)4-7-36(8-5-21)20(37)39-19(23(28,29)30)24(31,32)33/h1-2,13,19H,3-12,14-15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280490
PNG
(US10030020, Example 35 | US10781211, Example 204)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(cc(c2)C(F)(F)F)N2CCOCC2)CC1)C(F)(F)F
Show InChI InChI=1S/C24H28F9N3O3/c25-22(26,27)17-12-16(13-18(14-17)34-8-10-38-11-9-34)15-36-5-1-2-21(36)3-6-35(7-4-21)20(37)39-19(23(28,29)30)24(31,32)33/h12-14,19H,1-11,15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280491
PNG
(US10030020, Example 36 | US10781211, Example 203)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(cc(c2)C(F)(F)F)N2CCCC2)CC1)C(F)(F)F
Show InChI InChI=1S/C24H28F9N3O2/c25-22(26,27)17-12-16(13-18(14-17)34-7-1-2-8-34)15-36-9-3-4-21(36)5-10-35(11-6-21)20(37)38-19(23(28,29)30)24(31,32)33/h12-14,19H,1-11,15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280492
PNG
(US10030020, Example 37 | US10781211, Example 37)
Show SMILES FC(F)(F)Oc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)N1CCOCC1
Show InChI InChI=1S/C24H28F9N3O4/c25-22(26,27)19(23(28,29)30)39-20(37)35-6-3-21(4-7-35)2-1-5-36(21)15-16-12-17(34-8-10-38-11-9-34)14-18(13-16)40-24(31,32)33/h12-14,19H,1-11,15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280500
PNG
(US10030020, Example 45 | US10781211, Example 45)
Show SMILES FC1CCN(CC1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F
Show InChI InChI=1S/C25H29F10N3O2/c26-18-2-8-36(9-3-18)19-13-16(12-17(14-19)23(27,28)29)15-38-7-1-4-22(38)5-10-37(11-6-22)21(39)40-20(24(30,31)32)25(33,34)35/h12-14,18,20H,1-11,15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280502
PNG
(US10030020, Example 47 | US10781211, Example 47)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(cc(c2)C(F)(F)F)N2CCC2)CC1)C(F)(F)F
Show InChI InChI=1S/C23H26F9N3O2/c24-21(25,26)16-11-15(12-17(13-16)33-6-2-7-33)14-35-8-1-3-20(35)4-9-34(10-5-20)19(36)37-18(22(27,28)29)23(30,31)32/h11-13,18H,1-10,14H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280505
PNG
(US10030020, Example 50 | US10781211, Example 50)
Show SMILES CC1(C)CC2(CN1Cc1ccc(Cl)cc1N1CCOCC1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F
Show InChI InChI=1S/C25H32ClF6N3O3/c1-22(2)15-23(5-7-34(8-6-23)21(36)38-20(24(27,28)29)25(30,31)32)16-35(22)14-17-3-4-18(26)13-19(17)33-9-11-37-12-10-33/h3-4,13,20H,5-12,14-16H2,1-2H3
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280516
PNG
(US10030020, Example 61 | US10781211, Example 61)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(Cl)c2)CC1)C(F)(F)F
Show InChI InChI=1S/C19H21ClF6N2O2/c20-14-4-1-3-13(11-14)12-28-8-2-5-17(28)6-9-27(10-7-17)16(29)30-15(18(21,22)23)19(24,25)26/h1,3-4,11,15H,2,5-10,12H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280529
PNG
(US10030020, Example 74 | US10781211, Example 74)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2N2CCCCC2)CC1)C(F)(F)F
Show InChI InChI=1S/C24H30ClF6N3O2/c25-18-6-5-17(19(15-18)32-10-2-1-3-11-32)16-34-12-4-7-22(34)8-13-33(14-9-22)21(35)36-20(23(26,27)28)24(29,30)31/h5-6,15,20H,1-4,7-14,16H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280535
PNG
(US10030020, Example 80 | US10781211, Example 80)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3CCCCC3)c2Cl)CC1)C(F)(F)F
Show InChI InChI=1S/C24H30ClF6N3O2/c25-19-17(6-4-7-18(19)32-11-2-1-3-12-32)16-34-13-5-8-22(34)9-14-33(15-10-22)21(35)36-20(23(26,27)28)24(29,30)31/h4,6-7,20H,1-3,5,8-16H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280547
PNG
(US10030020, Example 92 | US10781211, Example 92)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(cc2N2CCS(=O)(=O)CC2)C(F)(F)F)CC1)C(F)(F)F
Show InChI InChI=1S/C24H28F9N3O4S/c25-22(26,27)17-3-2-16(18(14-17)34-10-12-41(38,39)13-11-34)15-36-7-1-4-21(36)5-8-35(9-6-21)20(37)40-19(23(28,29)30)24(31,32)33/h2-3,14,19H,1,4-13,15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280566
PNG
(US10030020, Example 111 | US10781211, Example 111)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3CCC(F)(F)CC3)c2Cl)CC1)C(F)(F)F
Show InChI InChI=1S/C24H28ClF8N3O2/c25-18-16(3-1-4-17(18)34-13-8-22(26,27)9-14-34)15-36-10-2-5-21(36)6-11-35(12-7-21)20(37)38-19(23(28,29)30)24(31,32)33/h1,3-4,19H,2,5-15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280571
PNG
(US10030020, Example 116 | US10781211, Example 116)
Show SMILES CCN1CCN(CC1)c1cccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1Cl
Show InChI InChI=1S/C25H33ClF6N4O2/c1-2-33-13-15-34(16-14-33)19-6-3-5-18(20(19)26)17-36-10-4-7-23(36)8-11-35(12-9-23)22(37)38-21(24(27,28)29)25(30,31)32/h3,5-6,21H,2,4,7-17H2,1H3
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride lipase


(Homo sapiens (Human))
BDBM280577
PNG
(US10030020, Example 122 | US10781211, Example 122)
Show SMILES OC(=O)C1CCN(CC1)c1cc(Cl)cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1
Show InChI InChI=1S/C25H30ClF6N3O4/c26-18-12-16(13-19(14-18)33-8-2-17(3-9-33)20(36)37)15-35-7-1-4-23(35)5-10-34(11-6-23)22(38)39-21(24(27,28)29)25(30,31)32/h12-14,17,21H,1-11,15H2,(H,36,37)
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
Human: Proteomes (human prefrontal cortex or cell membrane fractions) (50 μL, 1.0-2.0 mg/mL total protein concentration) were preincubated with ...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride lipase


(Homo sapiens (Human))
BDBM280578
PNG
(US10030020, Example 123 | US10781211, Example 123)
Show SMILES OC(=O)C1CCN(CC1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F
Show InChI InChI=1S/C26H30F9N3O4/c27-24(28,29)18-12-16(13-19(14-18)36-8-2-17(3-9-36)20(39)40)15-38-7-1-4-23(38)5-10-37(11-6-23)22(41)42-21(25(30,31)32)26(33,34)35/h12-14,17,21H,1-11,15H2,(H,39,40)
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
Human: Proteomes (human prefrontal cortex or cell membrane fractions) (50 μL, 1.0-2.0 mg/mL total protein concentration) were preincubated with ...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280600
PNG
(US10030020, Example 145 | US10781211, Example 145)
Show SMILES CC(=O)N1CCc2cccc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c2C1
Show InChI InChI=1S/C24H29F6N3O3/c1-16(34)32-11-6-17-4-2-5-18(19(17)15-32)14-33-10-3-7-22(33)8-12-31(13-9-22)21(35)36-20(23(25,26)27)24(28,29)30/h2,4-5,20H,3,6-15H2,1H3
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280605
PNG
(US10030020, Example 150 | US10781211, Example 150)
Show SMILES CCc1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1F
Show InChI InChI=1S/C21H25F7N2O2/c1-2-15-12-14(4-5-16(15)22)13-30-9-3-6-19(30)7-10-29(11-8-19)18(31)32-17(20(23,24)25)21(26,27)28/h4-5,12,17H,2-3,6-11,13H2,1H3
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280625
PNG
(US10030020, Example 170 | US10781211, Example 170)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(OC3CCOCC3)cc(c2)C(F)(F)F)CC1)C(F)(F)F
Show InChI InChI=1S/C25H29F9N2O4/c26-23(27,28)17-12-16(13-19(14-17)39-18-2-10-38-11-3-18)15-36-7-1-4-22(36)5-8-35(9-6-22)21(37)40-20(24(29,30)31)25(32,33)34/h12-14,18,20H,1-11,15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride lipase


(Homo sapiens (Human))
BDBM280633
PNG
(US10030020, Example 178 | US10781211, Example 178)
Show SMILES NC(=O)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1C(F)(F)F
Show InChI InChI=1S/C21H22F9N3O3/c22-19(23,24)14-3-2-12(10-13(14)15(31)34)11-33-7-1-4-18(33)5-8-32(9-6-18)17(35)36-16(20(25,26)27)21(28,29)30/h2-3,10,16H,1,4-9,11H2,(H2,31,34)
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
Human: Proteomes (human prefrontal cortex or cell membrane fractions) (50 μL, 1.0-2.0 mg/mL total protein concentration) were preincubated with ...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280639
PNG
(US10030020, Example 184 | US10781211, Example 184)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)c(c2)C(F)(F)F)CC1)C(F)(F)F
Show InChI InChI=1S/C20H20ClF9N2O2/c21-14-3-2-12(10-13(14)18(22,23)24)11-32-7-1-4-17(32)5-8-31(9-6-17)16(33)34-15(19(25,26)27)20(28,29)30/h2-3,10,15H,1,4-9,11H2
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US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride lipase


(Homo sapiens (Human))
BDBM463978
PNG
(US10781211, Example 202)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3cc(cc(c3)C(F)(F)F)N3CCCC3)C2)CC1)C(F)(F)F
Show InChI InChI=1S/C24H28F9N3O2/c25-22(26,27)17-11-16(12-18(13-17)35-6-1-2-7-35)14-34-8-3-21(15-34)4-9-36(10-5-21)20(37)38-19(23(28,29)30)24(31,32)33/h11-13,19H,1-10,14-15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
Human: Proteomes (human prefrontal cortex or cell membrane fractions) (50 μL, 1.0-2.0 mg/mL total protein concentration) were preincubated with ...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride lipase


(Homo sapiens (Human))
BDBM280662
PNG
(US10030020, Example 209 | US10781211, Example 209)
Show SMILES OC(=O)C1CN(CCO1)c1cc(ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F
Show InChI InChI=1S/C25H28F9N3O5/c26-23(27,28)16-2-1-15(17(11-16)37-9-10-41-18(13-37)19(38)39)12-35-6-3-22(14-35)4-7-36(8-5-22)21(40)42-20(24(29,30)31)25(32,33)34/h1-2,11,18,20H,3-10,12-14H2,(H,38,39)
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
Human: Proteomes (human prefrontal cortex or cell membrane fractions) (50 μL, 1.0-2.0 mg/mL total protein concentration) were preincubated with ...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride lipase


(Homo sapiens (Human))
BDBM280665
PNG
(US10030020, Example 214 | US10781211, Example 214)
Show SMILES OC(=O)[C@@H]1CCCN(C1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F
Show InChI InChI=1S/C26H30F9N3O4/c27-24(28,29)18-5-4-16(19(13-18)37-9-1-3-17(14-37)20(39)40)15-38-10-2-6-23(38)7-11-36(12-8-23)22(41)42-21(25(30,31)32)26(33,34)35/h4-5,13,17,21H,1-3,6-12,14-15H2,(H,39,40)/t17-/m1/s1
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
Human: Proteomes (human prefrontal cortex or cell membrane fractions) (50 μL, 1.0-2.0 mg/mL total protein concentration) were preincubated with ...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride lipase


(Homo sapiens (Human))
BDBM280678
PNG
(US10030020, Example 230 | US10781211, Example 230)
Show SMILES CC1(CCN(C1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F)C(O)=O
Show InChI InChI=1S/C26H30F9N3O4/c1-22(20(39)40)6-10-37(15-22)18-13-17(24(27,28)29)4-3-16(18)14-38-9-2-5-23(38)7-11-36(12-8-23)21(41)42-19(25(30,31)32)26(33,34)35/h3-4,13,19H,2,5-12,14-15H2,1H3,(H,39,40)
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
Human: Proteomes (human prefrontal cortex or cell membrane fractions) (50 μL, 1.0-2.0 mg/mL total protein concentration) were preincubated with ...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280460
PNG
(US10030020, Example 5 | US10781211, Example 5)
Show SMILES CCOc1cccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1
Show InChI InChI=1S/C21H26F6N2O3/c1-2-31-16-6-3-5-15(13-16)14-29-10-4-7-19(29)8-11-28(12-9-19)18(30)32-17(20(22,23)24)21(25,26)27/h3,5-6,13,17H,2,4,7-12,14H2,1H3
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280464
PNG
(US10030020, Example 9 | US10781211, Example 9)
Show SMILES COc1cc(Cl)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F
Show InChI InChI=1S/C20H23ClF6N2O3/c1-31-15-11-14(21)4-3-13(15)12-29-8-2-5-18(29)6-9-28(10-7-18)17(30)32-16(19(22,23)24)20(25,26)27/h3-4,11,16H,2,5-10,12H2,1H3
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280495
PNG
(US10030020, Example 40 | US10781211, Example 40)
Show SMILES CS(=O)(=O)N1CCN(CC1)c1cc(Cl)cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)c1
Show InChI InChI=1S/C24H31ClF6N4O4S/c1-40(37,38)35-11-9-32(10-12-35)19-14-17(13-18(25)15-19)16-34-6-2-3-22(34)4-7-33(8-5-22)21(36)39-20(23(26,27)28)24(29,30)31/h13-15,20H,2-12,16H2,1H3
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280496
PNG
(US10030020, Example 41 | US10781211, Example 41)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(cc(c2)C(F)(F)F)N2CCN(CC2)C2CC2)CC1)C(F)(F)F
Show InChI InChI=1S/C27H33F9N4O2/c28-25(29,30)19-14-18(15-21(16-19)38-12-10-37(11-13-38)20-2-3-20)17-40-7-1-4-24(40)5-8-39(9-6-24)23(41)42-22(26(31,32)33)27(34,35)36/h14-16,20,22H,1-13,17H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280498
PNG
(US10030020, Example 43 | US10781211, Example 43)
Show SMILES CS(=O)(=O)N1CCN(CC1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F
Show InChI InChI=1S/C25H31F9N4O4S/c1-43(40,41)38-11-9-35(10-12-38)19-14-17(13-18(15-19)23(26,27)28)16-37-6-2-3-22(37)4-7-36(8-5-22)21(39)42-20(24(29,30)31)25(32,33)34/h13-15,20H,2-12,16H2,1H3
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280506
PNG
(US10030020, Example 51 | US10781211, Example 51)
Show SMILES CC1(C)CC2(CN1Cc1ccc(cc1N1CCOCC1)C(F)(F)F)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F
Show InChI InChI=1S/C26H32F9N3O3/c1-22(2)15-23(5-7-37(8-6-23)21(39)41-20(25(30,31)32)26(33,34)35)16-38(22)14-17-3-4-18(24(27,28)29)13-19(17)36-9-11-40-12-10-36/h3-4,13,20H,5-12,14-16H2,1-2H3
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280517
PNG
(US10030020, Example 62 | US10781211, Example 62)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2)CC1)C(F)(F)F
Show InChI InChI=1S/C19H21ClF6N2O2/c20-14-4-2-13(3-5-14)12-28-9-1-6-17(28)7-10-27(11-8-17)16(29)30-15(18(21,22)23)19(24,25)26/h2-5,15H,1,6-12H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280526
PNG
(US10030020, Example 71 | US10781211, Example 71)
Show SMILES CCN1CCCc2cccc(CN3CCC4(C3)CCN(CC4)C(=O)OC(C(F)(F)F)C(F)(F)F)c12
Show InChI InChI=1S/C24H31F6N3O2/c1-2-32-11-4-7-17-5-3-6-18(19(17)32)15-31-12-8-22(16-31)9-13-33(14-10-22)21(34)35-20(23(25,26)27)24(28,29)30/h3,5-6,20H,2,4,7-16H2,1H3
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280531
PNG
(US10030020, Example 76 | US10781211, Example 76)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2ccc(Cl)cc2N2CCCC2)CC1)C(F)(F)F
Show InChI InChI=1S/C23H28ClF6N3O2/c24-17-5-4-16(18(14-17)31-9-1-2-10-31)15-33-11-3-6-21(33)7-12-32(13-8-21)20(34)35-19(22(25,26)27)23(28,29)30/h4-5,14,19H,1-3,6-13,15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280534
PNG
(US10030020, Example 79 | US10781211, Example 79)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3CCOCC3)c2Cl)CC1)C(F)(F)F
Show InChI InChI=1S/C23H28ClF6N3O3/c24-18-16(3-1-4-17(18)31-11-13-35-14-12-31)15-33-8-2-5-21(33)6-9-32(10-7-21)20(34)36-19(22(25,26)27)23(28,29)30/h1,3-4,19H,2,5-15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280537
PNG
(US10030020, Example 82 | US10781211, Example 82)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3CC4CCC(C3)O4)c2Cl)CC1)C(F)(F)F
Show InChI InChI=1S/C25H30ClF6N3O3/c26-20-16(3-1-4-19(20)34-14-17-5-6-18(15-34)37-17)13-35-10-2-7-23(35)8-11-33(12-9-23)22(36)38-21(24(27,28)29)25(30,31)32/h1,3-4,17-18,21H,2,5-15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280540
PNG
(US10030020, Example 85 | US10781211, Example 85)
Show SMILES Cc1c(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cccc1N1CCCC1
Show InChI InChI=1S/C24H31F6N3O2/c1-17-18(6-4-7-19(17)31-11-2-3-12-31)16-33-13-5-8-22(33)9-14-32(15-10-22)21(34)35-20(23(25,26)27)24(28,29)30/h4,6-7,20H,2-3,5,8-16H2,1H3
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280548
PNG
(US10030020, Example 93 | US10781211, Example 93)
Show SMILES CC(=O)NC1CCN(CC1)c1cc(ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F
Show InChI InChI=1S/C27H33F9N4O3/c1-17(41)37-20-5-11-38(12-6-20)21-15-19(25(28,29)30)4-3-18(21)16-40-10-2-7-24(40)8-13-39(14-9-24)23(42)43-22(26(31,32)33)27(34,35)36/h3-4,15,20,22H,2,5-14,16H2,1H3,(H,37,41)
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280557
PNG
(US10030020, Example 102 | US10781211, Example 102)
Show SMILES FC1CCN(CC1)c1cc(Cl)ccc1CN1CCCC11CCN(CC1)C(=O)OC(C(F)(F)F)C(F)(F)F
Show InChI InChI=1S/C24H29ClF7N3O2/c25-17-3-2-16(19(14-17)33-10-4-18(26)5-11-33)15-35-9-1-6-22(35)7-12-34(13-8-22)21(36)37-20(23(27,28)29)24(30,31)32/h2-3,14,18,20H,1,4-13,15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280564
PNG
(US10030020, Example 109 | US10781211, Example 109)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3C4CCC3COC4)c2Cl)CC1)C(F)(F)F
Show InChI InChI=1S/C25H30ClF6N3O3/c26-20-16(3-1-4-19(20)35-17-5-6-18(35)15-37-14-17)13-34-10-2-7-23(34)8-11-33(12-9-23)22(36)38-21(24(27,28)29)25(30,31)32/h1,3-4,17-18,21H,2,5-15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280569
PNG
(US10030020, Example 114 | US10781211, Example 114)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cccc(N3CCN(CC=O)CC3)c2Cl)CC1)C(F)(F)F
Show InChI InChI=1S/C25H31ClF6N4O3/c26-20-18(3-1-4-19(20)34-13-11-33(12-14-34)15-16-37)17-36-8-2-5-23(36)6-9-35(10-7-23)22(38)39-21(24(27,28)29)25(30,31)32/h1,3-4,16,21H,2,5-15,17H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280598
PNG
(US10030020, Example 143 | US10781211, Example 143)
Show SMILES CS(=O)(=O)N1CCCc2cccc(CN3CCCC33CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)c12
Show InChI InChI=1S/C23H29F6N3O4S/c1-37(34,35)32-12-3-7-16-5-2-6-17(18(16)32)15-31-11-4-8-21(31)9-13-30(14-10-21)20(33)36-19(22(24,25)26)23(27,28)29/h2,5-6,19H,3-4,7-15H2,1H3
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280612
PNG
(US10030020, Example 157 | US10781211, Example 157)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCN(Cc3ccc(c(c3)N3CCCC3)C(F)(F)F)C2)CC1)C(F)(F)F
Show InChI InChI=1S/C24H28F9N3O2/c25-22(26,27)17-4-3-16(13-18(17)35-8-1-2-9-35)14-34-10-5-21(15-34)6-11-36(12-7-21)20(37)38-19(23(28,29)30)24(31,32)33/h3-4,13,19H,1-2,5-12,14-15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280631
PNG
(US10030020, Example 176 | US10781211, Example 176)
Show SMILES FC(F)(F)C(OC(=O)N1CCC2(CCCN2Cc2cc(OC3CCS(=O)(=O)CC3)cc(c2)C(F)(F)F)CC1)C(F)(F)F
Show InChI InChI=1S/C25H29F9N2O5S/c26-23(27,28)17-12-16(13-19(14-17)40-18-2-10-42(38,39)11-3-18)15-36-7-1-4-22(36)5-8-35(9-6-22)21(37)41-20(24(29,30)31)25(32,33)34/h12-14,18,20H,1-11,15H2
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280633
PNG
(US10030020, Example 178 | US10781211, Example 178)
Show SMILES NC(=O)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1C(F)(F)F
Show InChI InChI=1S/C21H22F9N3O3/c22-19(23,24)14-3-2-12(10-13(14)15(31)34)11-33-7-1-4-18(33)5-8-32(9-6-18)17(35)36-16(20(25,26)27)21(28,29)30/h2-3,10,16H,1,4-9,11H2,(H2,31,34)
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride lipase


(Homo sapiens (Human))
BDBM280634
PNG
(US10030020, Example 179 | US10781211, Example 179)
Show SMILES OC(=O)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)ccc1C(F)(F)F
Show InChI InChI=1S/C21H21F9N2O4/c22-19(23,24)14-3-2-12(10-13(14)15(33)34)11-32-7-1-4-18(32)5-8-31(9-6-18)17(35)36-16(20(25,26)27)21(28,29)30/h2-3,10,16H,1,4-9,11H2,(H,33,34)
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
Human: Proteomes (human prefrontal cortex or cell membrane fractions) (50 μL, 1.0-2.0 mg/mL total protein concentration) were preincubated with ...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280637
PNG
(US10030020, Example 182 | US10781211, Example 182)
Show SMILES OC(=O)c1ccc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc1C(F)(F)F
Show InChI InChI=1S/C21H21F9N2O4/c22-19(23,24)14-10-12(2-3-13(14)15(33)34)11-32-7-1-4-18(32)5-8-31(9-6-18)17(35)36-16(20(25,26)27)21(28,29)30/h2-3,10,16H,1,4-9,11H2,(H,33,34)
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride Lipase (MGL)


(Mus musculus (mouse))
BDBM280647
PNG
(US10030020, Example 192 | US10781211, Example 192)
Show SMILES CC1(C)CC2(CN1Cc1cc(CN3CCOCC3)ccc1OC(F)(F)F)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F
Show InChI InChI=1S/C27H34F9N3O4/c1-23(2)16-24(5-7-38(8-6-24)22(40)42-21(25(28,29)30)26(31,32)33)17-39(23)15-19-13-18(14-37-9-11-41-12-10-37)3-4-20(19)43-27(34,35)36/h3-4,13,21H,5-12,14-17H2,1-2H3
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
MAGL, ABHD6 and FAAH: Proteomes (mouse brain membrane fraction or cell lysates) (50 μL, 1.0 mg/mL total protein concentration) were preincubated...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride lipase


(Homo sapiens (Human))
BDBM463988
PNG
(US10781211, Example 216)
Show SMILES CC1CCCN(C1)c1cc(ccc1CN1CCC2(C1)CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)C(F)(F)F
Show InChI InChI=1S/C26H32F9N3O2/c1-17-3-2-9-38(14-17)20-13-19(24(27,28)29)5-4-18(20)15-36-10-6-23(16-36)7-11-37(12-8-23)22(39)40-21(25(30,31)32)26(33,34)35/h4-5,13,17,21H,2-3,6-12,14-16H2,1H3
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
Human: Proteomes (human prefrontal cortex or cell membrane fractions) (50 μL, 1.0-2.0 mg/mL total protein concentration) were preincubated with ...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride lipase


(Homo sapiens (Human))
BDBM280673
PNG
(US10030020, Example 223 | US10781211, Example 223)
Show SMILES CC1(CCCN(C1)c1cc(CN2CCC3(C2)CCN(CC3)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F)C(O)=O
Show InChI InChI=1S/C27H32F9N3O4/c1-23(21(40)41)3-2-7-39(15-23)19-12-17(11-18(13-19)25(28,29)30)14-37-8-4-24(16-37)5-9-38(10-6-24)22(42)43-20(26(31,32)33)27(34,35)36/h11-13,20H,2-10,14-16H2,1H3,(H,40,41)
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
Human: Proteomes (human prefrontal cortex or cell membrane fractions) (50 μL, 1.0-2.0 mg/mL total protein concentration) were preincubated with ...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
Monoglyceride lipase


(Homo sapiens (Human))
BDBM464000
PNG
(US10781211, Example 231)
Show SMILES CC1CCN(C1)c1cc(CN2CCCC22CCN(CC2)C(=O)OC(C(F)(F)F)C(F)(F)F)cc(c1)C(F)(F)F
Show InChI InChI=1S/C25H30F9N3O2/c1-16-3-8-36(14-16)19-12-17(11-18(13-19)23(26,27)28)15-37-7-2-4-22(37)5-9-35(10-6-22)21(38)39-20(24(29,30)31)25(32,33)34/h11-13,16,20H,2-10,14-15H2,1H3
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LUNDBECK LA JOLLA RESEARCH CENTER, INC.

US Patent


Assay Description
Human: Proteomes (human prefrontal cortex or cell membrane fractions) (50 μL, 1.0-2.0 mg/mL total protein concentration) were preincubated with ...


US Patent US10781211 (2020)

More data for this
Ligand-Target Pair
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* indicates data uncertainty>20%