Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with all data for entry = 9417
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM385387((E)-3-Fluoro-2-[[2-(4-methoxy-1-piperidyl)pyrimidi...)
Affinity DataIC50:  12nMAssay Description:Amine oxidase activity of recombinant SSAO, MAOa, and MAOb isoforms are measured using the MAO-Glo™ assay kit from Promega (V1402). Test compounds (w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM385388((E)-3-Fluoro-2-[[2-[(3S)-3-methoxypyrrolidin-1-yl]...)
Affinity DataIC50:  32nMAssay Description:Amine oxidase activity of recombinant SSAO, MAOa, and MAOb isoforms are measured using the MAO-Glo™ assay kit from Promega (V1402). Test compounds (w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM385389((3 S)-1-[5-[(E)-2-(Aminomethyl)-3-fluoro-allyloxy]...)
Affinity DataIC50:  52nMAssay Description:Amine oxidase activity of recombinant SSAO, MAOa, and MAOb isoforms are measured using the MAO-Glo™ assay kit from Promega (V1402). Test compounds (w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent