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Found 14 Enz. Inhib. hit(s) with all data for entry = 9451
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Aclaris Therapeutics

US Patent
LigandPNGBDBM466940(US10800775, Example 20 | propyl (R)-4-(1-(2-cyano-...)
Affinity DataIC50: <10nMAssay Description:The activity of JAK3 (a.a. 781-1124, ThermoFisher) was quantified by measuring the phosphorylation of SRCtide (FAM-GEEPLYWSFPAKKK-NH2). Kinase reacti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Aclaris Therapeutics

US Patent
LigandPNGBDBM466936(US10800775, Example 16 | ethyl 4-(1-(2-cyano-1-cyc...)
Affinity DataIC50: <10nMAssay Description:The activity of JAK3 (a.a. 781-1124, ThermoFisher) was quantified by measuring the phosphorylation of SRCtide (FAM-GEEPLYWSFPAKKK-NH2). Kinase reacti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Aclaris Therapeutics

US Patent
LigandPNGBDBM466934(US10800775, Example 1 | ethyl 4-(1-(2-cyano-1-cycl...)
Affinity DataIC50: <10nMAssay Description:The activity of JAK3 (a.a. 781-1124, ThermoFisher) was quantified by measuring the phosphorylation of SRCtide (FAM-GEEPLYWSFPAKKK-NH2). Kinase reacti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Aclaris Therapeutics

US Patent
LigandPNGBDBM466935(US10800775, Example 9 | ethyl 4-(1-(3-(cyanomethyl...)
Affinity DataIC50: <10nMAssay Description:The activity of JAK3 (a.a. 781-1124, ThermoFisher) was quantified by measuring the phosphorylation of SRCtide (FAM-GEEPLYWSFPAKKK-NH2). Kinase reacti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Aclaris Therapeutics

US Patent
LigandPNGBDBM466938(US10800775, Example 18 | isopropyl 4-(1-(2-cyano-1...)
Affinity DataIC50: <10nMAssay Description:The activity of JAK3 (a.a. 781-1124, ThermoFisher) was quantified by measuring the phosphorylation of SRCtide (FAM-GEEPLYWSFPAKKK-NH2). Kinase reacti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3 [781-1124](Homo sapiens (Human))
Aclaris Therapeutics

US Patent
LigandPNGBDBM466938(US10800775, Example 18 | isopropyl 4-(1-(2-cyano-1...)
Affinity DataIC50:  55nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Aclaris Therapeutics

US Patent
LigandPNGBDBM466939(US10800775, Example 19 | isopropyl 4-(1-(2-cyano-1...)
Affinity DataIC50:  55nMAssay Description:The activity of JAK3 (a.a. 781-1124, ThermoFisher) was quantified by measuring the phosphorylation of SRCtide (FAM-GEEPLYWSFPAKKK-NH2). Kinase reacti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3 [781-1124](Homo sapiens (Human))
Aclaris Therapeutics

US Patent
LigandPNGBDBM466939(US10800775, Example 19 | isopropyl 4-(1-(2-cyano-1...)
Affinity DataIC50:  55nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3 [781-1124](Homo sapiens (Human))
Aclaris Therapeutics

US Patent
LigandPNGBDBM466937(US10800775, Example 17 | ethyl 4-(1-(2-cyano-1-cyc...)
Affinity DataIC50:  55nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3 [781-1124](Homo sapiens (Human))
Aclaris Therapeutics

US Patent
LigandPNGBDBM466940(US10800775, Example 20 | propyl (R)-4-(1-(2-cyano-...)
Affinity DataIC50:  55nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3 [781-1124](Homo sapiens (Human))
Aclaris Therapeutics

US Patent
LigandPNGBDBM466936(US10800775, Example 16 | ethyl 4-(1-(2-cyano-1-cyc...)
Affinity DataIC50:  55nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3 [781-1124](Homo sapiens (Human))
Aclaris Therapeutics

US Patent
LigandPNGBDBM466935(US10800775, Example 9 | ethyl 4-(1-(3-(cyanomethyl...)
Affinity DataIC50:  55nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3 [781-1124](Homo sapiens (Human))
Aclaris Therapeutics

US Patent
LigandPNGBDBM466934(US10800775, Example 1 | ethyl 4-(1-(2-cyano-1-cycl...)
Affinity DataIC50:  55nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Aclaris Therapeutics

US Patent
LigandPNGBDBM466937(US10800775, Example 17 | ethyl 4-(1-(2-cyano-1-cyc...)
Affinity DataIC50:  55nMAssay Description:The activity of JAK3 (a.a. 781-1124, ThermoFisher) was quantified by measuring the phosphorylation of SRCtide (FAM-GEEPLYWSFPAKKK-NH2). Kinase reacti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent