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Patent code US10807956

Compile Data Set for Download or QSAR

Found 210 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314104
PNG
(3-{[4-(trifluoromethyl)benzyl]amino}pyridine-4-car...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(cc1)C(F)(F)F
Show InChI InChI=1S/C14H11F3N2O2/c15-14(16,17)10-3-1-9(2-4-10)7-19-12-8-18-6-5-11(12)13(20)21/h1-6,8,19H,7H2,(H,20,21)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314108
PNG
(3-[(4-phenoxybenzyl)amino]pyridine-4-carboxylic ac...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(Oc2ccccc2)cc1
Show InChI InChI=1S/C19H16N2O3/c22-19(23)17-10-11-20-13-18(17)21-12-14-6-8-16(9-7-14)24-15-4-2-1-3-5-15/h1-11,13,21H,12H2,(H,22,23)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314109
PNG
(3-({2-[(dimethylamino)methyl]benzyl}amino)pyridine...)
Show SMILES CN(C)Cc1ccccc1CNc1cnccc1C(O)=O
Show InChI InChI=1S/C16H19N3O2/c1-19(2)11-13-6-4-3-5-12(13)9-18-15-10-17-8-7-14(15)16(20)21/h3-8,10,18H,9,11H2,1-2H3,(H,20,21)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314110
PNG
(3-[(3,4-dichlorobenzyl)amino]pyridine-4-carboxylic...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(Cl)c(Cl)c1
Show InChI InChI=1S/C13H10Cl2N2O2/c14-10-2-1-8(5-11(10)15)6-17-12-7-16-4-3-9(12)13(18)19/h1-5,7,17H,6H2,(H,18,19)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314116
PNG
(3-[(4-chloro-2-methoxybenzyl)amino]pyridine-4-carb...)
Show SMILES COc1cc(Cl)ccc1CNc1cnccc1C(O)=O
Show InChI InChI=1S/C14H13ClN2O3/c1-20-13-6-10(15)3-2-9(13)7-17-12-8-16-5-4-11(12)14(18)19/h2-6,8,17H,7H2,1H3,(H,18,19)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314117
PNG
(3-[(4-chloro-2-hydroxybenzyl)amino]pyridine-4-carb...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(Cl)cc1O
Show InChI InChI=1S/C13H11ClN2O3/c14-9-2-1-8(12(17)5-9)6-16-11-7-15-4-3-10(11)13(18)19/h1-5,7,16-17H,6H2,(H,18,19)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314118
PNG
(3-[(2-aminobenzyl)amino]pyridine-4-carboxylic acid...)
Show SMILES Nc1ccccc1CNc1cnccc1C(O)=O
Show InChI InChI=1S/C13H13N3O2/c14-11-4-2-1-3-9(11)7-16-12-8-15-6-5-10(12)13(17)18/h1-6,8,16H,7,14H2,(H,17,18)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314119
PNG
(3-[(4-bromobenzyl)amino]pyridine-4-carboxylic acid...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(Br)cc1
Show InChI InChI=1S/C13H11BrN2O2/c14-10-3-1-9(2-4-10)7-16-12-8-15-6-5-11(12)13(17)18/h1-6,8,16H,7H2,(H,17,18)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314122
PNG
(3-[(4-chloro-2-cyclopropylbenzyl)amino]pyridine-4-...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(Cl)cc1C1CC1
Show InChI InChI=1S/C16H15ClN2O2/c17-12-4-3-11(14(7-12)10-1-2-10)8-19-15-9-18-6-5-13(15)16(20)21/h3-7,9-10,19H,1-2,8H2,(H,20,21)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314122
PNG
(3-[(4-chloro-2-cyclopropylbenzyl)amino]pyridine-4-...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(Cl)cc1C1CC1
Show InChI InChI=1S/C16H15ClN2O2/c17-12-4-3-11(14(7-12)10-1-2-10)8-19-15-9-18-6-5-13(15)16(20)21/h3-7,9-10,19H,1-2,8H2,(H,20,21)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314126
PNG
(3-[(2-cyclopropyl-3-methylbenzyl)amino]pyridine-4-...)
Show SMILES Cc1cccc(CNc2cnccc2C(O)=O)c1C1CC1
Show InChI InChI=1S/C17H18N2O2/c1-11-3-2-4-13(16(11)12-5-6-12)9-19-15-10-18-8-7-14(15)17(20)21/h2-4,7-8,10,12,19H,5-6,9H2,1H3,(H,20,21)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314127
PNG
(3-{[(4-cyclopropylpyridin-3-yl)-methyl]amino}pyrid...)
Show SMILES OC(=O)c1ccncc1NCc1cnccc1C1CC1
Show InChI InChI=1S/C15H15N3O2/c19-15(20)13-4-6-17-9-14(13)18-8-11-7-16-5-3-12(11)10-1-2-10/h3-7,9-10,18H,1-2,8H2,(H,19,20)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314130
PNG
(3-[(2-cyclopropyl-5-methylbenzyl)amino]pyridine-4-...)
Show SMILES Cc1ccc(C2CC2)c(CNc2cnccc2C(O)=O)c1
Show InChI InChI=1S/C17H18N2O2/c1-11-2-5-14(12-3-4-12)13(8-11)9-19-16-10-18-7-6-15(16)17(20)21/h2,5-8,10,12,19H,3-4,9H2,1H3,(H,20,21)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314136
PNG
(3-{[(5-methylfuran-2-yl)methyl]amino}pyridine-4-ca...)
Show SMILES Cc1ccc(CNc2cnccc2C(O)=O)o1
Show InChI InChI=1S/C12H12N2O3/c1-8-2-3-9(17-8)6-14-11-7-13-5-4-10(11)12(15)16/h2-5,7,14H,6H2,1H3,(H,15,16)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 4C


(Homo sapiens (Human))
BDBM314136
PNG
(3-{[(5-methylfuran-2-yl)methyl]amino}pyridine-4-ca...)
Show SMILES Cc1ccc(CNc2cnccc2C(O)=O)o1
Show InChI InChI=1S/C12H12N2O3/c1-8-2-3-9(17-8)6-14-11-7-13-5-4-10(11)12(15)16/h2-5,7,14H,6H2,1H3,(H,15,16)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314140
PNG
(3-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]p...)
Show SMILES OC(=O)c1ccncc1NCC1COc2ccccc2O1
Show InChI InChI=1S/C15H14N2O4/c18-15(19)11-5-6-16-8-12(11)17-7-10-9-20-13-3-1-2-4-14(13)21-10/h1-6,8,10,17H,7,9H2,(H,18,19)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 4C


(Homo sapiens (Human))
BDBM314140
PNG
(3-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]p...)
Show SMILES OC(=O)c1ccncc1NCC1COc2ccccc2O1
Show InChI InChI=1S/C15H14N2O4/c18-15(19)11-5-6-16-8-12(11)17-7-10-9-20-13-3-1-2-4-14(13)21-10/h1-6,8,10,17H,7,9H2,(H,18,19)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314141
PNG
(3-[(2,3-dihydro-1H-inden-1-ylmethylbenzyl)amino]py...)
Show SMILES OC(=O)c1ccncc1NCC1CCc2ccccc12
Show InChI InChI=1S/C16H16N2O2/c19-16(20)14-7-8-17-10-15(14)18-9-12-6-5-11-3-1-2-4-13(11)12/h1-4,7-8,10,12,18H,5-6,9H2,(H,19,20)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314141
PNG
(3-[(2,3-dihydro-1H-inden-1-ylmethylbenzyl)amino]py...)
Show SMILES OC(=O)c1ccncc1NCC1CCc2ccccc12
Show InChI InChI=1S/C16H16N2O2/c19-16(20)14-7-8-17-10-15(14)18-9-12-6-5-11-3-1-2-4-13(11)12/h1-4,7-8,10,12,18H,5-6,9H2,(H,19,20)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314156
PNG
(3-{[(6-methyl-3,4-dihydro-2H-chromen-4-yl)methyl]a...)
Show SMILES Cc1ccc2OCCC(CNc3cnccc3C(O)=O)c2c1
Show InChI InChI=1S/C17H18N2O3/c1-11-2-3-16-14(8-11)12(5-7-22-16)9-19-15-10-18-6-4-13(15)17(20)21/h2-4,6,8,10,12,19H,5,7,9H2,1H3,(H,20,21)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 4C


(Homo sapiens (Human))
BDBM314100
PNG
(3-[(4-fluorobenzyl)amino]pyridine-4-carboxylic aci...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(F)cc1
Show InChI InChI=1S/C13H11FN2O2/c14-10-3-1-9(2-4-10)7-16-12-8-15-6-5-11(12)13(17)18/h1-6,8,16H,7H2,(H,17,18)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314105
PNG
(3-[(biphenyl-4-ylmethyl)amino]pyridine-4-carboxyli...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(cc1)-c1ccccc1
Show InChI InChI=1S/C19H16N2O2/c22-19(23)17-10-11-20-13-18(17)21-12-14-6-8-16(9-7-14)15-4-2-1-3-5-15/h1-11,13,21H,12H2,(H,22,23)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314106
PNG
(3-[(4-chlorobenzyl)amino]pyridine-4-carboxylic aci...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(Cl)cc1
Show InChI InChI=1S/C13H11ClN2O2/c14-10-3-1-9(2-4-10)7-16-12-8-15-6-5-11(12)13(17)18/h1-6,8,16H,7H2,(H,17,18)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314111
PNG
(3-[(4-chloro-2-methylbenzyl)amino]pyridine-4-carbo...)
Show SMILES Cc1cc(Cl)ccc1CNc1cnccc1C(O)=O
Show InChI InChI=1S/C14H13ClN2O2/c1-9-6-11(15)3-2-10(9)7-17-13-8-16-5-4-12(13)14(18)19/h2-6,8,17H,7H2,1H3,(H,18,19)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314115
PNG
(3-[(2-cyclopropylbenzyl)amino]pyridine-4-carboxyli...)
Show SMILES OC(=O)c1ccncc1NCc1ccccc1C1CC1
Show InChI InChI=1S/C16H16N2O2/c19-16(20)14-7-8-17-10-15(14)18-9-12-3-1-2-4-13(12)11-5-6-11/h1-4,7-8,10-11,18H,5-6,9H2,(H,19,20)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 4C


(Homo sapiens (Human))
BDBM314115
PNG
(3-[(2-cyclopropylbenzyl)amino]pyridine-4-carboxyli...)
Show SMILES OC(=O)c1ccncc1NCc1ccccc1C1CC1
Show InChI InChI=1S/C16H16N2O2/c19-16(20)14-7-8-17-10-15(14)18-9-12-3-1-2-4-13(12)11-5-6-11/h1-4,7-8,10-11,18H,5-6,9H2,(H,19,20)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314121
PNG
(3-[(4-cyclopropylbenzyl)amino]pyridine-4-carboxyli...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(cc1)C1CC1
Show InChI InChI=1S/C16H16N2O2/c19-16(20)14-7-8-17-10-15(14)18-9-11-1-3-12(4-2-11)13-5-6-13/h1-4,7-8,10,13,18H,5-6,9H2,(H,19,20)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 4C


(Homo sapiens (Human))
BDBM314124
PNG
(3-[(naphthalene-1-ylmethyl)amino]pyridine-4-carbox...)
Show SMILES OC(=O)c1ccncc1NCc1cccc2ccccc12
Show InChI InChI=1S/C17H14N2O2/c20-17(21)15-8-9-18-11-16(15)19-10-13-6-3-5-12-4-1-2-7-14(12)13/h1-9,11,19H,10H2,(H,20,21)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314125
PNG
(3-[(1H-indol-7-ylmethyl)amino]pyridine-4-carboxyli...)
Show SMILES OC(=O)c1ccncc1NCc1cccc2cc[nH]c12
Show InChI InChI=1S/C15H13N3O2/c19-15(20)12-5-6-16-9-13(12)18-8-11-3-1-2-10-4-7-17-14(10)11/h1-7,9,17-18H,8H2,(H,19,20)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314128
PNG
(3-{[3-(trifluoromethyl)benzyl]amino}pyridine-4-car...)
Show SMILES OC(=O)c1ccncc1NCc1cccc(c1)C(F)(F)F
Show InChI InChI=1S/C14H11F3N2O2/c15-14(16,17)10-3-1-2-9(6-10)7-19-12-8-18-5-4-11(12)13(20)21/h1-6,8,19H,7H2,(H,20,21)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314134
PNG
(3-[(1-benzofuran-3-ylmethyl)amino]pyridine-4-carbo...)
Show SMILES OC(=O)c1ccncc1NCc1coc2ccccc12
Show InChI InChI=1S/C15H12N2O3/c18-15(19)12-5-6-16-8-13(12)17-7-10-9-20-14-4-2-1-3-11(10)14/h1-6,8-9,17H,7H2,(H,18,19)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314156
PNG
(3-{[(6-methyl-3,4-dihydro-2H-chromen-4-yl)methyl]a...)
Show SMILES Cc1ccc2OCCC(CNc3cnccc3C(O)=O)c2c1
Show InChI InChI=1S/C17H18N2O3/c1-11-2-3-16-14(8-11)12(5-7-22-16)9-19-15-10-18-6-4-13(15)17(20)21/h2-4,6,8,10,12,19H,5,7,9H2,1H3,(H,20,21)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 4C


(Homo sapiens (Human))
BDBM314158
PNG
(3-{[(6-fluoro-3,4-dihydro-2H-chromen-4-yl)methyl]a...)
Show SMILES OC(=O)c1ccncc1NCC1CCOc2cc(F)ccc12
Show InChI InChI=1S/C16H15FN2O3/c17-11-1-2-12-10(4-6-22-15(12)7-11)8-19-14-9-18-5-3-13(14)16(20)21/h1-3,5,7,9-10,19H,4,6,8H2,(H,20,21)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 4C


(Homo sapiens (Human))
BDBM314097
PNG
(3-(benzylamino)pyridazine-4-carboxylic acid | US10...)
Show SMILES OC(=O)c1ccnnc1NCc1ccccc1
Show InChI InChI=1S/C12H11N3O2/c16-12(17)10-6-7-14-15-11(10)13-8-9-4-2-1-3-5-9/h1-7H,8H2,(H,13,15)(H,16,17)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 4C


(Homo sapiens (Human))
BDBM314102
PNG
(3-{[4-hydroxymethyl)benzyl]amino}pyridine-4-carbox...)
Show SMILES OCc1ccc(CNc2cnccc2C(O)=O)cc1
Show InChI InChI=1S/C14H14N2O3/c17-9-11-3-1-10(2-4-11)7-16-13-8-15-6-5-12(13)14(18)19/h1-6,8,16-17H,7,9H2,(H,18,19)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314104
PNG
(3-{[4-(trifluoromethyl)benzyl]amino}pyridine-4-car...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(cc1)C(F)(F)F
Show InChI InChI=1S/C14H11F3N2O2/c15-14(16,17)10-3-1-9(2-4-10)7-19-12-8-18-6-5-11(12)13(20)21/h1-6,8,19H,7H2,(H,20,21)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314113
PNG
(3-[(2-hydroxybenzyl)amino]pyridine-4-carboxylic ac...)
Show SMILES OC(=O)c1ccncc1NCc1ccccc1O
Show InChI InChI=1S/C13H12N2O3/c16-12-4-2-1-3-9(12)7-15-11-8-14-6-5-10(11)13(17)18/h1-6,8,15-16H,7H2,(H,17,18)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314114
PNG
(3-[(2,4-dichlorobenzyl)amino]pyridine-4-carboxylic...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(Cl)cc1Cl
Show InChI InChI=1S/C13H10Cl2N2O2/c14-9-2-1-8(11(15)5-9)6-17-12-7-16-4-3-10(12)13(18)19/h1-5,7,17H,6H2,(H,18,19)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314117
PNG
(3-[(4-chloro-2-hydroxybenzyl)amino]pyridine-4-carb...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(Cl)cc1O
Show InChI InChI=1S/C13H11ClN2O3/c14-9-2-1-8(12(17)5-9)6-16-11-7-15-4-3-10(11)13(18)19/h1-5,7,16-17H,6H2,(H,18,19)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 4C


(Homo sapiens (Human))
BDBM314118
PNG
(3-[(2-aminobenzyl)amino]pyridine-4-carboxylic acid...)
Show SMILES Nc1ccccc1CNc1cnccc1C(O)=O
Show InChI InChI=1S/C13H13N3O2/c14-11-4-2-1-3-9(11)7-16-12-8-15-6-5-10(12)13(17)18/h1-6,8,16H,7,14H2,(H,17,18)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 4C


(Homo sapiens (Human))
BDBM314119
PNG
(3-[(4-bromobenzyl)amino]pyridine-4-carboxylic acid...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(Br)cc1
Show InChI InChI=1S/C13H11BrN2O2/c14-10-3-1-9(2-4-10)7-16-12-8-15-6-5-11(12)13(17)18/h1-6,8,16H,7H2,(H,17,18)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314120
PNG
(3-[(4-methylbenzyl)amino]pyridine-4-carboxylic aci...)
Show SMILES Cc1ccc(CNc2cnccc2C(O)=O)cc1
Show InChI InChI=1S/C14H14N2O2/c1-10-2-4-11(5-3-10)8-16-13-9-15-7-6-12(13)14(17)18/h2-7,9,16H,8H2,1H3,(H,17,18)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314123
PNG
(3-{[2-cyclopropyl-4-(trifluoromethyl)benzyl]amino}...)
Show SMILES OC(=O)c1ccncc1NCc1ccc(cc1C1CC1)C(F)(F)F
Show InChI InChI=1S/C17H15F3N2O2/c18-17(19,20)12-4-3-11(14(7-12)10-1-2-10)8-22-15-9-21-6-5-13(15)16(23)24/h3-7,9-10,22H,1-2,8H2,(H,23,24)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314132
PNG
(3-{[2-(phenylamino)benzyl]amino}pyridine-4-carboxy...)
Show SMILES OC(=O)c1ccncc1NCc1ccccc1Nc1ccccc1
Show InChI InChI=1S/C19H17N3O2/c23-19(24)16-10-11-20-13-18(16)21-12-14-6-4-5-9-17(14)22-15-7-2-1-3-8-15/h1-11,13,21-22H,12H2,(H,23,24)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314133
PNG
(3-{[3-(cyclopropylmethoxy)benzyl]amino}pyridine-4-...)
Show SMILES OC(=O)c1ccncc1NCc1cccc(OCC2CC2)c1
Show InChI InChI=1S/C17H18N2O3/c20-17(21)15-6-7-18-10-16(15)19-9-13-2-1-3-14(8-13)22-11-12-4-5-12/h1-3,6-8,10,12,19H,4-5,9,11H2,(H,20,21)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 4C


(Homo sapiens (Human))
BDBM50153334
PNG
(CHEMBL3774545 | US10179769, Example 39 | US1080795...)
Show SMILES Cc1ccc(CNc2cnccc2C(O)=O)s1
Show InChI InChI=1S/C12H12N2O2S/c1-8-2-3-9(17-8)6-14-11-7-13-5-4-10(11)12(15)16/h2-5,7,14H,6H2,1H3,(H,15,16)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314142
PNG
(3-[(1,2,3,4-tetrahydronaphthalen-1-ylmethyl)amino]...)
Show SMILES OC(=O)c1ccncc1NCC1CCCc2ccccc12
Show InChI InChI=1S/C17H18N2O2/c20-17(21)15-8-9-18-11-16(15)19-10-13-6-3-5-12-4-1-2-7-14(12)13/h1-2,4,7-9,11,13,19H,3,5-6,10H2,(H,20,21)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5B


(Homo sapiens (Human))
BDBM314142
PNG
(3-[(1,2,3,4-tetrahydronaphthalen-1-ylmethyl)amino]...)
Show SMILES OC(=O)c1ccncc1NCC1CCCc2ccccc12
Show InChI InChI=1S/C17H18N2O2/c20-17(21)15-8-9-18-11-16(15)19-10-13-6-3-5-12-4-1-2-7-14(12)13/h1-2,4,7-9,11,13,19H,3,5-6,10H2,(H,20,21)
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n/an/a<100n/an/an/an/an/an/a



CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of Jarid1B was determined in 384 well plate format under the following reaction conditions: 0.8...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314154
PNG
(3-{[(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)m...)
Show SMILES COc1ccc2C(CNc3cnccc3C(O)=O)CCCc2c1
Show InChI InChI=1S/C18H20N2O3/c1-23-14-5-6-15-12(9-14)3-2-4-13(15)10-20-17-11-19-8-7-16(17)18(21)22/h5-9,11,13,20H,2-4,10H2,1H3,(H,21,22)
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CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
Lysine-specific demethylase 5A


(Homo sapiens (Human))
BDBM314097
PNG
(3-(benzylamino)pyridazine-4-carboxylic acid | US10...)
Show SMILES OC(=O)c1ccnnc1NCc1ccccc1
Show InChI InChI=1S/C12H11N3O2/c16-12(17)10-6-7-14-15-11(10)13-8-9-4-2-1-3-5-9/h1-7H,8H2,(H,13,15)(H,16,17)
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n/an/a<100n/an/an/an/an/an/a



CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...


US Patent US10807956 (2020)

More data for this
Ligand-Target Pair
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* indicates data uncertainty>20%