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Found 32 Enz. Inhib. hit(s) with all data for entry = 9592
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476253( (Z)-ethyl 5-(4-((tert-butyldimethylsilyl)oxy)-3-m...)
Affinity DataKi:  0.780nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476252(2-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6...)
Affinity DataKi:  1.01nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476251((R)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiaz...)
Affinity DataKi:  1.42nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476249(4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6...)
Affinity DataKi:  1.57nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

US Patent
LigandPNGBDBM50392121(CHEMBL2152632 | US10874669, Compound (+-)-10)
Affinity DataKi:  1.92nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

US Patent
LigandPNGBDBM50392123(CHEMBL2152634 | US10874669, Compound (-)-10)
Affinity DataKi:  2.19nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476250(US10874669, Compound 34 (D-575))
Affinity DataKi:  2.59nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476248(US10874669, Compound 23 (D-548))
Affinity DataKi:  3.62nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

US Patent
LigandPNGBDBM476245(6-((2-(4-(4-chloro-1H-indol-5-yl)piperazin-1-yl)et...)
Affinity DataKi:  10.4nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476256(4-(3-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6...)
Affinity DataKi:  11.9nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476260((S)-5-(4-(4-(2-((2-amino-4,5,6,7-tetrahydrobenzo[d...)
Affinity DataKi:  14.2nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476247(4-(3-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6...)
Affinity DataKi:  15.8nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Wayne State University

US Patent
LigandPNGBDBM50392122(CHEMBL2152633 | US10874669, Compound (+)-10)
Affinity DataKi:  15.9nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476254((Z)-4-(5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiaz...)
Affinity DataKi:  23.3nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476255((Z)-4-(5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiaz...)
Affinity DataKi:  25nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wayne State University

US Patent
LigandPNGBDBM50392123(CHEMBL2152634 | US10874669, Compound (-)-10)
Affinity DataKi:  39nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476257((E)-4-(3-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiaz...)
Affinity DataKi:  39.1nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wayne State University

US Patent
LigandPNGBDBM50392121(CHEMBL2152632 | US10874669, Compound (+-)-10)
Affinity DataKi:  46.7nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476251((R)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiaz...)
Affinity DataKi:  65.7nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476249(4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6...)
Affinity DataKi:  68.3nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wayne State University

US Patent
LigandPNGBDBM476245(6-((2-(4-(4-chloro-1H-indol-5-yl)piperazin-1-yl)et...)
Affinity DataKi:  76.4nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476253( (Z)-ethyl 5-(4-((tert-butyldimethylsilyl)oxy)-3-m...)
Affinity DataKi:  112nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476250(US10874669, Compound 34 (D-575))
Affinity DataKi:  116nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476252(2-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6...)
Affinity DataKi:  117nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476255((Z)-4-(5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiaz...)
Affinity DataKi:  121nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wayne State University

US Patent
LigandPNGBDBM50392122(CHEMBL2152633 | US10874669, Compound (+)-10)
Affinity DataKi:  134nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476260((S)-5-(4-(4-(2-((2-amino-4,5,6,7-tetrahydrobenzo[d...)
Affinity DataKi:  162nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476248(US10874669, Compound 23 (D-548))
Affinity DataKi:  175nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476254((Z)-4-(5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiaz...)
Affinity DataKi:  233nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476256(4-(3-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6...)
Affinity DataKi:  499nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476247(4-(3-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6...)
Affinity DataKi:  2.40E+3nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wayne State University

US Patent
LigandPNGBDBM476257((E)-4-(3-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiaz...)
Affinity DataKi:  4.63E+3nMAssay Description:A well established radioligand competition assay was carried out to evaluate binding affinity of the test compounds and were compared with that of th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent