Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 9629
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Topivert Pharma

US Patent
LigandPNGBDBM477065(US10882859, Reference compound PF-06263276)
Affinity DataKd:  2.70nMAssay Description:The biochemical JAK family enzyme binding assays carried out at DiscoveRx.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Topivert Pharma

US Patent
LigandPNGBDBM477065(US10882859, Reference compound PF-06263276)
Affinity DataKd:  0.780nMAssay Description:The biochemical JAK family enzyme binding assays carried out at DiscoveRx.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Topivert Pharma

US Patent
LigandPNGBDBM477065(US10882859, Reference compound PF-06263276)
Affinity DataKd:  1.90nMAssay Description:The biochemical JAK family enzyme binding assays carried out at DiscoveRx.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Topivert Pharma

US Patent
LigandPNGBDBM477065(US10882859, Reference compound PF-06263276)
Affinity DataKd:  1.90nMAssay Description:The biochemical JAK family enzyme binding assays carried out at DiscoveRx.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Topivert Pharma

US Patent
LigandPNGBDBM477066(US10882859, Example 1)
Affinity DataKd:  0.620nMAssay Description:The biochemical JAK family enzyme binding assays carried out at DiscoveRx.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Topivert Pharma

US Patent
LigandPNGBDBM477067(US10882859, Example 2(a))
Affinity DataKd:  0.0690nMAssay Description:The biochemical JAK family enzyme binding assays carried out at DiscoveRx.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Topivert Pharma

US Patent
LigandPNGBDBM477066(US10882859, Example 1)
Affinity DataKd:  0.0980nMAssay Description:The biochemical JAK family enzyme binding assays carried out at DiscoveRx.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Topivert Pharma

US Patent
LigandPNGBDBM477066(US10882859, Example 1)
Affinity DataKd:  0.110nMAssay Description:The biochemical JAK family enzyme binding assays carried out at DiscoveRx.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Topivert Pharma

US Patent
LigandPNGBDBM477067(US10882859, Example 2(a))
Affinity DataKd:  0.600nMAssay Description:The biochemical JAK family enzyme binding assays carried out at DiscoveRx.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Topivert Pharma

US Patent
LigandPNGBDBM477067(US10882859, Example 2(a))
Affinity DataKd:  0.0340nMAssay Description:The biochemical JAK family enzyme binding assays carried out at DiscoveRx.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Topivert Pharma

US Patent
LigandPNGBDBM477067(US10882859, Example 2(a))
Affinity DataKd:  0.0460nMAssay Description:The biochemical JAK family enzyme binding assays carried out at DiscoveRx.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Topivert Pharma

US Patent
LigandPNGBDBM477066(US10882859, Example 1)
Affinity DataKd:  0.0520nMAssay Description:The biochemical JAK family enzyme binding assays carried out at DiscoveRx.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent