Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 9674
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dana Farber Cancer Institute

US Patent
LigandPNGBDBM480781(US10906878, Compound 84A)
Affinity DataIC50:  3.12nMAssay Description:1. Optimization of kinase concentration required to determine ATP Km,app. The assay was first performed at a high concentration of ATP (1 mM) against...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dana Farber Cancer Institute

US Patent
LigandPNGBDBM480780(US10906878, Compound 83A)
Affinity DataIC50:  5.13nMAssay Description:1. Optimization of kinase concentration required to determine ATP Km,app. The assay was first performed at a high concentration of ATP (1 mM) against...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dana Farber Cancer Institute

US Patent
LigandPNGBDBM480782(US10906878, Compound 85A)
Affinity DataIC50:  5.74nMAssay Description:1. Optimization of kinase concentration required to determine ATP Km,app. The assay was first performed at a high concentration of ATP (1 mM) against...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dana Farber Cancer Institute

US Patent
LigandPNGBDBM480777(US10906878, Compound 29A)
Affinity DataIC50:  19.4nMAssay Description:1. Optimization of kinase concentration required to determine ATP Km,app. The assay was first performed at a high concentration of ATP (1 mM) against...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dana Farber Cancer Institute

US Patent
LigandPNGBDBM480776(US10906878, Compound 25A)
Affinity DataIC50:  31.2nMAssay Description:1. Optimization of kinase concentration required to determine ATP Km,app. The assay was first performed at a high concentration of ATP (1 mM) against...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dana Farber Cancer Institute

US Patent
LigandPNGBDBM480778(US10906878, Compound 103A)
Affinity DataIC50:  2.24E+3nMAssay Description:1. Optimization of kinase concentration required to determine ATP Km,app. The assay was first performed at a high concentration of ATP (1 mM) against...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dana Farber Cancer Institute

US Patent
LigandPNGBDBM480779(US10906878, Compound 104A)
Affinity DataIC50: >1.00E+4nMAssay Description:1. Optimization of kinase concentration required to determine ATP Km,app. The assay was first performed at a high concentration of ATP (1 mM) against...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent