Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 9694
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM155363(US10383871, Example 9 | US10918640, Example 9 | US...)
Affinity DataIC50:  3nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM155368(US10383871, Example 15 | US10918640, Example 15 | ...)
Affinity DataIC50:  7nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM155359(US10383871, Example 5 | US10918640, Example 5 | US...)
Affinity DataIC50:  9nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM155372(US10383871, Example 17 | US10918640, Example 17 | ...)
Affinity DataIC50:  12nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM155366(US10383871, Example 12 | US10918640, Example 12 | ...)
Affinity DataIC50:  12nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM482174(3-[5-(2,6-Difluoro-phenyl)-pyridin-2-yloxy]-azetid...)
Affinity DataIC50:  14nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM482174(3-[5-(2,6-Difluoro-phenyl)-pyridin-2-yloxy]-azetid...)
Affinity DataIC50:  16nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM155362(US10383871, Example 8 | US10918640, Example 8 | US...)
Affinity DataIC50:  18nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM155361(US10383871, Example 7 | US10918640, Example 7 | US...)
Affinity DataIC50:  19nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM155365(US10383871, Example 11 | US10918640, Example 11 | ...)
Affinity DataIC50:  19nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM155369(US10383871, Example 19 | US10918640, Example 19 | ...)
Affinity DataIC50:  26nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM155367(US10383871, Example 13 | US10918640, Example 13 | ...)
Affinity DataIC50:  38nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM155371(US10383871, Example 16 | US10918640, Example 16 | ...)
Affinity DataIC50:  42nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM155364(US10383871, Example 10 | US10918640, Example 10 | ...)
Affinity DataIC50:  49nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Vernalis (R&D)

US Patent
LigandPNGBDBM155358(US10383871, Example 4 | US10918640, Example 4 | US...)
Affinity DataIC50:  67nMAssay Description:Active rat FAAH protein (30-579) was isolated as described in the literature. The coding sequence of amino adds 30-579 of rat FAAH were cloned into t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM155360(US10383871, Example 6 | US10918640, Example 6 | US...)
Affinity DataIC50:  73nMAssay Description:Human FAAH 1 activity was determined by measuring the liberation of the highly fluorescent 7-amino, 4-methyl Coumarin (AMC) generated during hydrolys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Vernalis (R&D)

US Patent
LigandPNGBDBM155357(US10383871, Example 3 | US10918640, Example 3 | US...)
Affinity DataIC50:  77nMAssay Description:Active rat FAAH protein (30-579) was isolated as described in the literature. The coding sequence of amino adds 30-579 of rat FAAH were cloned into t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Vernalis (R&D)

US Patent
LigandPNGBDBM155355(US10383871, Example 1 | US10918640, Example 1 | US...)
Affinity DataIC50:  135nMAssay Description:Active rat FAAH protein (30-579) was isolated as described in the literature. The coding sequence of amino adds 30-579 of rat FAAH were cloned into t...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Vernalis (R&D)

US Patent
LigandPNGBDBM155356(US10383871, Example 2 | US10918640, Example 2 | US...)
Affinity DataIC50:  279nMAssay Description:Active rat FAAH protein (30-579) was isolated as described in the literature. The coding sequence of amino adds 30-579 of rat FAAH were cloned into t...More data for this Ligand-Target Pair
In DepthDetails US Patent