Compile Data Set for Download or QSAR
maximum 50k data
Found 1210 Enz. Inhib. hit(s) with all data for entry = 9956
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503258((2R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(4-cyan...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503260((2R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-[4-cyan...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503263((2R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-2-methyl-...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503264((2R,6S)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-2,6-di...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503265((2R,6S)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(3-c...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503266(N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-[5- (trifluo...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503271((2R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(2,6-di...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503272((2R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-[4-cyan...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503273((2R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(4-cyan...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503277((2R,6R)-4-[4-amino-5-(trifluoromethyl)pyrimidin-2-...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503278((2R,6R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(5-c...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503280((2R,6R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-2,6-di...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503281((2R,6R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-2,6-di...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503282((2R,6R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-2,6-di...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503122(N-[(2S)-2-(1-benzylpiperidin-4-yl)-2-hydroxyethyl]...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503143((3R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-1-(5-cyan...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503144((3R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-3-methyl-...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503145((3R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-1-[3-fluo...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503188(N-[2-(1-benzylpiperidin-4-yl)ethyl]-7-methyl-2-[3-...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503190(N-[2-(1-benzyl-4-hydroxypiperidin-4-yl)ethyl]-7-me...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503192(N-[(2S)-2-(1-benzylpiperidin-4-yl)-2-hydroxyethyl]...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503193(N-[(2R)-2-(1-benzylpiperidin-4-yl)-2-hydroxyethyl]...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503196(N-[2-(1-benzylpiperidin-4-yl)ethyl]-2-(2,4-difluor...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503199(N-[2-(1-benzylpiperidin-4-yl)ethyl]-2-(4-fluorophe...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503200(N-[2-(1-benzylpiperidin-4-yl)ethyl]-2-(3,5-difluor...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503211(N-[2-(1-benzylpiperidin-4-yl)ethyl]-7-methyl-2-[3-...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503212(N-[2-(1-benzylpiperidin-4-yl)ethyl]-7-methyl-2-(3,...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503225((3R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-3-methyl-...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503226((3R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-1-(5-chlo...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM502819((2S,6R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(5-c...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503233((2R,6S)-4-(5-cyanopyrimidin-2-yl)-2,6-dimethyl-N-(...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503240((2R)-2-methyl-N-(2-{1-[alpha,alpha-2H-benzyl]piper...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM502819((2S,6R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(5-c...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503242((2R)-4-[4-amino-5-(trifluoromethyl)pyrimidin-2-yl]...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503242((2R)-4-[4-amino-5-(trifluoromethyl)pyrimidin-2-yl]...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503245((2R,6S)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(4-c...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503246((2R,6S)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(4-c...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503247((2R,6S)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(4-c...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503248((2R,6S)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(3,5...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503250((2R,6S)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(3-c...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503251((2R,6S)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(6-c...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503252((2R,6S)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(4-c...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503253((2R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(4-cyan...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503255((2R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(4-cyan...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503256((2R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(4-chlo...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503257((2R)-N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(4-chlo...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503051(N-{2-[1-benzyl-3-(hydroxymethyl)piperidin-4-yl]eth...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503052(N-[2-(1-benzylpiperidin-4-yl)ethyl]-1-[3-chloro-5 ...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM503053(N-{2-[1-benzyl-4-(hydroxymethyl)piperidin-4-yl]eth...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Neurocrine Biosciences

US Patent
LigandPNGBDBM502996(N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-[4- (trifluo...)
Affinity DataKi: <10nMAssay Description:Binding affinity (Ki) of compounds was measured by inhibition of radioligand binding to membranes from CHO cells expressing human M1, M2, M3, M4 and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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