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Found 14 Enz. Inhib. hit(s) with all data for entry = 7607
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Amitech Therapeutic Solutions

US Patent
LigandPNGBDBM205483(US9260417, 6)
Affinity DataKd:  52nMAssay Description:For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Amitech Therapeutic Solutions

US Patent
LigandPNGBDBM205483(US9260417, 6)
Affinity DataKd:  170nMAssay Description:For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Amitech Therapeutic Solutions

US Patent
LigandPNGBDBM205483(US9260417, 6)
Affinity DataKd:  300nMAssay Description:For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Amitech Therapeutic Solutions

US Patent
LigandPNGBDBM205483(US9260417, 6)
Affinity DataKd:  520nMAssay Description:For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase-like 2(Homo sapiens (Human))
Amitech Therapeutic Solutions

US Patent
LigandPNGBDBM205483(US9260417, 6)
Affinity DataKd:  5.10E+3nMAssay Description:For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCyclin-dependent kinase 11B(Homo sapiens (Human))
Amitech Therapeutic Solutions

US Patent
LigandPNGBDBM205483(US9260417, 6)
Affinity DataKd:  7.50E+3nMAssay Description:For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Amitech Therapeutic Solutions

US Patent
LigandPNGBDBM205483(US9260417, 6)
Affinity DataKd: >1.00E+4nMAssay Description:For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Amitech Therapeutic Solutions

US Patent
LigandPNGBDBM205483(US9260417, 6)
Affinity DataKd: >1.00E+4nMAssay Description:For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Amitech Therapeutic Solutions

US Patent
LigandPNGBDBM205483(US9260417, 6)
Affinity DataKd: >1.00E+4nMAssay Description:For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Amitech Therapeutic Solutions

US Patent
LigandPNGBDBM205483(US9260417, 6)
Affinity DataKd: >1.00E+4nMAssay Description:For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Amitech Therapeutic Solutions

US Patent
LigandPNGBDBM205483(US9260417, 6)
Affinity DataKd: >1.00E+4nMAssay Description:For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Amitech Therapeutic Solutions

US Patent
LigandPNGBDBM205483(US9260417, 6)
Affinity DataKd: >1.00E+4nMAssay Description:For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Amitech Therapeutic Solutions

US Patent
LigandPNGBDBM205483(US9260417, 6)
Affinity DataKd: >1.00E+4nMAssay Description:For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Amitech Therapeutic Solutions

US Patent
LigandPNGBDBM205483(US9260417, 6)
Affinity DataKd: >1.00E+4nMAssay Description:For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEsc...More data for this Ligand-Target Pair
In DepthDetails US Patent