Compile Data Set for Download or QSAR
maximum 50k data
Found 41 Enz. Inhib. hit(s) with all data for entry = 7590
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204888(US9260454, 21)
Affinity DataIC50:  14nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204894(US9260454, 28)
Affinity DataIC50:  45nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204910(US9260454, 69)
Affinity DataIC50:  54nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204897(US9260454, 38)
Affinity DataIC50:  61nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204911(US9260454, 70)
Affinity DataIC50:  62nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204895(US9260454, 29)
Affinity DataIC50:  62nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204909(US9260454, 68)
Affinity DataIC50:  65nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204922(US9260454, 89)
Affinity DataIC50:  72nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204887(US9260454, 20)
Affinity DataIC50:  110nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204914(US9260454, 78)
Affinity DataIC50:  120nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204900(US9260454, 44)
Affinity DataIC50:  120nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204913(US9260454, 74)
Affinity DataIC50:  130nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204902(US9260454, 46)
Affinity DataIC50:  140nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204915(US9260454, 80)
Affinity DataIC50:  150nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204908(US9260454, 63 | US9260454, 85)
Affinity DataIC50:  200nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204899(US9260454, 42)
Affinity DataIC50:  240nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204921(US9260454, 88)
Affinity DataIC50:  250nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204884(US9260454, 5)
Affinity DataIC50:  270nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204898(US9260454, 40)
Affinity DataIC50:  340nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204892(US9260454, 26)
Affinity DataIC50:  340nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204891(US9260454, 24)
Affinity DataIC50:  370nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204893(US9260454, 27)
Affinity DataIC50:  420nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204896(US9260454, 36)
Affinity DataIC50:  430nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204917(US9260454, 83)
Affinity DataIC50:  750nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204890(US9260454, 23)
Affinity DataIC50:  800nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204906(US9260454, 59)
Affinity DataIC50:  1.00E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204882(US9260454, 6)
Affinity DataIC50:  1.10E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204912(US9260454, 72)
Affinity DataIC50:  1.20E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204889(US9260454, 22)
Affinity DataIC50:  1.40E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204904(US9260454, 53)
Affinity DataIC50:  1.70E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204919(US9260454, 84)
Affinity DataIC50:  1.70E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204905(US9260454, 55)
Affinity DataIC50:  2.00E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204918(US9260454, 86)
Affinity DataIC50:  2.10E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204903(US9260454, 50)
Affinity DataIC50:  2.30E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204908(US9260454, 63 | US9260454, 85)
Affinity DataIC50:  2.60E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204916(US9260454, 81)
Affinity DataIC50:  2.90E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204907(US9260454, 62)
Affinity DataIC50:  3.10E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204901(US9260454, 45)
Affinity DataIC50:  4.30E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204885(US9260454, 10)
Affinity DataIC50:  1.20E+4nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204883(US9260454, 8)
Affinity DataIC50:  1.80E+4nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM204886(US9260454, 16)
Affinity DataIC50:  2.60E+4nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent