Found 4 Enz. Inhib. hit(s) with all data for entry = 8159 
Affinity DataIC50: 1.70nMpH: 7.4 T: 2°CAssay Description:The assay was performed using Kinase-Glo Plus luminescence kinase assay kit (Promega). The compounds were diluted in 10% DMSO and 5 μl of the dilu...More data for this Ligand-Target Pair
Affinity DataIC50: <10nMpH: 7.4 T: 2°CAssay Description:The assay was performed using Kinase-Glo Plus luminescence kinase assay kit (Promega). The compounds were diluted in 10% DMSO and 5 μl of the dilu...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor [668-1210,T790M,L858R](Homo sapiens (Human))
Teligene
US Patent
Teligene
US Patent
Affinity DataIC50: 22nMpH: 7.4 T: 2°CAssay Description:The assay was performed using Kinase-Glo Plus luminescence kinase assay kit (Promega). The compounds were diluted in 10% DMSO and 5 μl of the dilu...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor [668-1210,T790M,L858R](Homo sapiens (Human))
Teligene
US Patent
Teligene
US Patent
Affinity DataIC50: <100nMpH: 7.4 T: 2°CAssay Description:The assay was performed using Kinase-Glo Plus luminescence kinase assay kit (Promega). The compounds were diluted in 10% DMSO and 5 μl of the dilu...More data for this Ligand-Target Pair
