Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 1330
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratories Del Dr. Esteve

US Patent
LigandPNGBDBM317225(6-(Azepan-1- ylmethyl)-2- phenylimidazo[2,1- b]thi...)
Affinity DataKi:  16nMAssay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratories Del Dr. Esteve

US Patent
LigandPNGBDBM317227(6-((2-(Azepan-1- ylethoxy)methyl)-2- phenylimidazo...)
Affinity DataKi:  40nMAssay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratories Del Dr. Esteve

US Patent
LigandPNGBDBM317226(6-((4- Methylpiperazin-1- ylmethyl)-2- phenylimida...)
Affinity DataKi:  56nMAssay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratories Del Dr. Esteve

US Patent
LigandPNGBDBM317230(2-(Azepan-1- ylmethyl)-6- phenylimidazo[2,1- b]thi...)
Affinity DataKi:  100nMAssay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratories Del Dr. Esteve

US Patent
LigandPNGBDBM317218(US9617281, Compound 4)
Affinity DataKi:  168nMAssay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratories Del Dr. Esteve

US Patent
LigandPNGBDBM317228(2-Phenyl-6-((2- (pyrrolidin-1- yl)ethoxy)methyl) i...)
Affinity DataKi:  190nMAssay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratories Del Dr. Esteve

US Patent
LigandPNGBDBM317231(2-(4-Fluorophenyl)- 6-((4- methylpiperazin-1- yl)m...)
Affinity DataKi:  210nMAssay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Laboratories Del Dr. Esteve

US Patent
LigandPNGBDBM317229(6-((4- Methylpiperazin-1- ylmethyl)-2- phenylimida...)
Affinity DataKi:  260nMAssay Description:Brain membrane preparation and binding assays for the σ1-receptor were performed as described (DeHaven-Hudkins, D. L., L. C. Fleissner, and F. Y...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent