Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 2632
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373532(US9903855, Molecule 1)
Affinity DataIC50:  440nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373534(US9903855, Molecule 2)
Affinity DataIC50:  500nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373536(US9903855, Molecule 3)
Affinity DataIC50:  640nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373537(US9903855, Molecule 4)
Affinity DataIC50:  670nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373532(US9903855, Molecule 1)
Affinity DataIC50:  770nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373538(US9903855, Molecule 5)
Affinity DataIC50:  870nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373536(US9903855, Molecule 3)
Affinity DataIC50:  8.76E+3nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373536(US9903855, Molecule 3)
Affinity DataIC50: >1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373538(US9903855, Molecule 5)
Affinity DataIC50: >1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373536(US9903855, Molecule 3)
Affinity DataIC50: >1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373537(US9903855, Molecule 4)
Affinity DataIC50: >1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373537(US9903855, Molecule 4)
Affinity DataIC50: >1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373537(US9903855, Molecule 4)
Affinity DataIC50: >1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373538(US9903855, Molecule 5)
Affinity DataIC50: >1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373538(US9903855, Molecule 5)
Affinity DataIC50: >1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373534(US9903855, Molecule 2)
Affinity DataIC50: >1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373534(US9903855, Molecule 2)
Affinity DataIC50: >1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373532(US9903855, Molecule 1)
Affinity DataIC50: >1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373532(US9903855, Molecule 1)
Affinity DataIC50: >1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
The Regents Of The University Of California

US Patent
LigandPNGBDBM373534(US9903855, Molecule 2)
Affinity DataIC50: >1.00E+4nMAssay Description:Please see Hutti, et al., (2012). Development of a High-Throughput Assay for Identifying Inhibitors of TBK1 and IKKε.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent