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Found 2 Enz. Inhib. hit(s) for PDB: 1JLQ
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Glaxosmithkline

LigandPNGBDBM1802(2-Amino-6-arylthiobenzonitrile deriv. 3v, 739W94 |...)
Affinity DataIC50:  7nMAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
University Of Perugia

Curated by ChEMBL
LigandPNGBDBM1802(2-Amino-6-arylthiobenzonitrile deriv. 3v, 739W94 |...)
Affinity DataIC50:  7.10nMAssay Description:Inhibitory concentration against Reverse transcriptaseMore data for this Ligand-Target Pair