Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) for PDB: 2XK8
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50330576(4-(3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl)...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of NEK2 autophosphorylation after 2 hrs by DELFIA assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50330576(4-(3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl)...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of NEK2 by microfluidic assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50330576(4-(3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl)...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of NEK2 assessed as inhibition of substrate phosphorylationMore data for this Ligand-Target Pair