Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) for PDB: 2XKC
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50330577(4-(3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl)...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of NEK2 assessed as inhibition of substrate phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50330577(4-(3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl)...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of NEK2 assessed as inhibition of substrate phosphorylationMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50330577(4-(3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl)...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of NEK2 by microfluidic assayMore data for this Ligand-Target Pair