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Found 2 Enz. Inhib. hit(s) for PDB: 3D4Q
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006650(CHEMBL526479)
Affinity DataIC50:  0.0300nMAssay Description:Inhibition of BRAF (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50006650(CHEMBL526479)
Affinity DataIC50:  9nMAssay Description:Inhibition of BRAF (unknown origin)-mediated ERK phosphorylationMore data for this Ligand-Target Pair