Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) for PDB: 3OT8
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334852(3-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-5-(piperi...)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant His-CHK1 expressed in baculovirus after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50334852(3-methyl-N-(3-(1-methyl-1H-pyrazol-4-yl)-5-(piperi...)
Affinity DataIC50:  9nMAssay Description:Inhibition of histidine-tagged recombinant CHK1 expressed in baculovirus expression system after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair