Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) for PDB: 3UP2
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM87051(Bisanilinopyrimidine inhibitor, 5 | Bisanilinopyri...)
Affinity DataIC50:  28nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM87051(Bisanilinopyrimidine inhibitor, 5 | Bisanilinopyri...)
Affinity DataIC50:  28nM Kd:  40nMpH: 7.4 T: 2°CAssay Description:The formation of ADP from ATP was quantified using a coupled enzyme assay (DiscoverX) in with a fluorescent resorufin dye is generated from the inter...More data for this Ligand-Target Pair