Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) for PDB: 4APU
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375437(CHEMBL409661)
Affinity DataIC50:  0.610nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375437(CHEMBL409661)
Affinity DataEC50:  0.660nMAssay Description:Agonist activity at human PRB expressed in CHO cellsMore data for this Ligand-Target Pair