Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) for PDB: 4DON
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399448(CHEMBL1230189)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of BRD4 isoform 1 by AlphaScreen assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399448(CHEMBL1230189)
Affinity DataKd:  3.89E+4nMAssay Description:Binding affinity to human His10-tagged BRD4 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 using 1% DMSO by SPR assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399448(CHEMBL1230189)
Affinity DataKd:  1.70E+4nMAssay Description:Binding affinity to human His10-tagged BRD4 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 using methanol by SPR assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399448(CHEMBL1230189)
Affinity DataKd:  2.04E+4nMAssay Description:Binding affinity to human His10-tagged BRD4 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 using 0.5% DMSO by SPR assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50399448(CHEMBL1230189)
Affinity DataKd:  1.02E+5nMAssay Description:Binding affinity to human His10-tagged BRD4 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 using 3% DMSO by SPR assayMore data for this Ligand-Target Pair