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Found 6 Enz. Inhib. hit(s) for PDB: 4FUC
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50138662(6-Carbamimidoyl-naphthalene-2-carboxylic acid (4-a...)
Affinity DataKi:  40nM ΔG°:  -42.2kJ/molepH: 7.4 T: 2°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
LigandPNGBDBM50138662(6-Carbamimidoyl-naphthalene-2-carboxylic acid (4-a...)
Affinity DataKi:  40nMAssay Description:Photometric_Method1More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50138662(6-Carbamimidoyl-naphthalene-2-carboxylic acid (4-a...)
Affinity DataKi:  40nMAssay Description:Inhibition of urokinaseMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50138662(6-Carbamimidoyl-naphthalene-2-carboxylic acid (4-a...)
Affinity DataKi:  40nMAssay Description:Binding affinity to human urokinase-type plasminogen activator (microPa).More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50138662(6-Carbamimidoyl-naphthalene-2-carboxylic acid (4-a...)
Affinity DataKi:  40nMAssay Description:Inhibition of human uPA using pyroGlu-Gly-Arg-p-NA.HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins by spectrop...More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Csar

LigandPNGBDBM50138662(6-Carbamimidoyl-naphthalene-2-carboxylic acid (4-a...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human uPA using pyroGlu-Gly-Arg-p-NA.HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins by spectrop...More data for this Ligand-Target Pair