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Found 3 Enz. Inhib. hit(s) for PDB: 4K9T
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of California Irvine

LigandPNGBDBM119125(GS4)
Affinity DataIC50:  1.50E+4nMAssay Description:The inhibitory potency of compounds GS4-GS8 on the 7-benzyloxy-4-(trifluoromethyl)coumarin hydroxylase activity of CYP3A4 was evaluated according to ...More data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of California Irvine

LigandPNGBDBM119125(GS4)
Affinity DataKd:  1.31E+4nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of California Irvine

LigandPNGBDBM119125(GS4)
Affinity DataKd:  1.50E+3nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair