Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) for PDB: 4MDQ
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Pittsburgh

US Patent
LigandPNGBDBM192239(US9187441, KK271)
Affinity DataKi:  900nM ΔG°:  -33.9kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Pittsburgh

US Patent
LigandPNGBDBM50014090(CHEMBL3260846)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of fluorescent P4 peptide from recombinant human MDM2 (18 to 125) expressed in Escherichia coli BL21(DE3) RIL expression system after 30...More data for this Ligand-Target Pair