Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) for PDB: 4NTX
TargetAcid-sensing ion channel 1(Rattus norvegicus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM16173(3,5-diamino-6-chloro-N-(diaminomethylene)pyrazinam...)
Affinity DataIC50:  3.02E+4nMAssay Description:Inhibition of ASIC1 in Sprague-Dawley rat articular chondrocytes assessed as decrease in acid-induced intracellular calcium level by Fluo-3AM dye bas...More data for this Ligand-Target Pair