Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) for PDB: 4Q1C
TargetDeoxycytidine kinase(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50440179(CHEMBL2426567)
Affinity DataKi:  2nMAssay Description:Apparent inhibition of human dCK by steady-state kinetic assayMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50440179(CHEMBL2426567)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of [3H]-dC uptake by scintillation counting analysisMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50440179(CHEMBL2426567)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50440179(CHEMBL2426567)
Affinity DataIC50:  18nMAssay Description:Apparent inhibition of human dCK assessed as phosphorylation activity by spectroscopic NADH-dependent enzyme-coupled assayMore data for this Ligand-Target Pair