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Compile Data Set for Download or QSAR
maximum 50k data
Found
1
Enz. Inhib. hit(s) for PDB:
5ACY
Target
Bromodomain-containing protein 4
(Homo sapiens (Human))
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50028128
(CHEMBL3353992)
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Affinity Data
IC50: 398nM
Assay Description:
Displacement of biotinylated tetra-acetylated histone H4 from His6-tagged BRD4 (1 to 477 aa) (unknown origin) after 1 hr by TR-FRET assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
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