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Found 5 Enz. Inhib. hit(s) for PDB: 5B0X
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50420563(CHEMBL2087023)
Affinity DataIC50:  11nMAssay Description:Inhibition of GST-tagged human CK2alpha' (1 to 350 residues) using CK2tide as substrate incubated for 1 hr by off-chip mobility shift assayMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50420563(CHEMBL2087023)
Affinity DataIC50:  20nMAssay Description:Inhibition of GST-tagged human CK2alpha (1 to 391 residues) using CK2tide as substrate incubated for 1 hr by off-chip mobility shift assayMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50420563(CHEMBL2087023)
Affinity DataIC50:  20nMAssay Description:Inhibition of human CK2alpha (2 to 391 residues) using [33P]-ATP by scintillation counting based radioactive filter binding assayMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50420563(CHEMBL2087023)
Affinity DataIC50:  32nMAssay Description:Competitive inhibition of GST fused human CK2alpha expressed in Escherichia coli BL21 after 10 mins in presence of ATPMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50420563(CHEMBL2087023)
Affinity DataIC50:  46nMAssay Description:Competitive inhibition of GST fused human CK2alpha' expressed in Escherichia coli BL21 after 10 mins in presence of ATPMore data for this Ligand-Target Pair