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Found 5 Enz. Inhib. hit(s) for PDB: 5LVR
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM152260(US8993552, 1F4 Compound 44)
Affinity DataKd:  1.08E+6nMAssay Description:Binding affinity to human His6-tagged PCAF expressed in Escherichia coli BL21(DE3)-R3 using 3% DMSO by SPR assayMore data for this Ligand-Target Pair
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM152260(US8993552, 1F4 Compound 44)
Affinity DataKd:  2.50E+5nMAssay Description:Binding affinity to human His6-tagged PCAF expressed in Escherichia coli BL21(DE3)-R3 using methanol by SPR assayMore data for this Ligand-Target Pair
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM152260(US8993552, 1F4 Compound 44)
Affinity DataKd:  2.50E+5nMAssay Description:Displacement of biotinylated small molecule ligand from His/FLAG-tagged PCAF bromodomain (719 to 832 residues) (unknown origin) after 15 mins by Alph...More data for this Ligand-Target Pair
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM152260(US8993552, 1F4 Compound 44)
Affinity DataKd:  3.60E+5nMAssay Description:Binding affinity to human His6-tagged PCAF expressed in Escherichia coli BL21(DE3)-R3 using 0.5% DMSO by SPR assayMore data for this Ligand-Target Pair
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
University Of Dundee

Curated by ChEMBL
LigandPNGBDBM152260(US8993552, 1F4 Compound 44)
Affinity DataKd:  6.60E+5nMAssay Description:Binding affinity to human His6-tagged PCAF expressed in Escherichia coli BL21(DE3)-R3 using 1% DMSO by SPR assayMore data for this Ligand-Target Pair