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Found 3 Enz. Inhib. hit(s) for PDB: 5YOJ
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50288363(CHEMBL4173216)
Affinity DataEC50:  25nMAssay Description:Inhibition of protease L10F/V32I/M46I/I47V/Q58E/I84V mutant in HIV1 A17 infected in human MT4 cells assessed as reduction in virus-induced cytopathic...More data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50288363(CHEMBL4173216)
Affinity DataEC50:  1.20nMAssay Description:Inhibition of DRV-resistant protease V32I/L33F/I54M/I84V mutant in HIV1 transfected in 293T cells after 48 hrs by lentiviral vector-based luciferase ...More data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50288363(CHEMBL4173216)
Affinity DataEC50:  0.300nMAssay Description:Inhibition of DRV-resistant protease V32I/L33F/I54M/V82I mutant in HIV1 transfected in 293T cells after 48 hrs by lentiviral vector-based luciferase ...More data for this Ligand-Target Pair