Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) for PDB: 5Z1S
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50465297(CHEMBL4283230)
Affinity DataIC50:  690nMAssay Description:Inhibition of human His6-tagged BRD4 BD1 (N44 to E168 residues) expressed in Escherichia coli BL21 (DE3) cells using H-SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50465297(CHEMBL4283230)
Affinity DataKd:  302nMAssay Description:Binding affinity to human His6-tagged BRD4 BD1 (N44 to E168 residues) expressed in Escherichia coli BL21 (DE3) cells by isothermal titration calorime...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB