Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) for PDB: 6C7R
TargetBromodomain-containing protein 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366670(CHEMBL4173488)
Affinity DataKi: <1nMAssay Description:Inhibition of FAM-labeled ZBA248 binding to recombinant human BRD4 bromodomain 1 (44 to 168 residues) expressed in Rosetta2 Escherichia coli DE3 cell...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366670(CHEMBL4173488)
Affinity DataIC50:  2nMAssay Description:Inhibition of FAM-labeled ZBA248 binding to recombinant human BRD4 bromodomain 1 (44 to 168 residues) expressed in Rosetta2 Escherichia coli DE3 cell...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366670(CHEMBL4173488)
Affinity DataKd:  2.20nMAssay Description:Binding affinity to human BRD4 bromodomain 1 (N44 to E168 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366670(CHEMBL4173488)
Affinity DataKd:  0.800nMAssay Description:Binding affinity to human BRD4 bromodomain 2 (K333 to E460 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair