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Found 32 Enz. Inhib. hit(s) with all data for entry = 50009897
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088982(CHEMBL160253 | CHEMBL367004 | N-[1-(1-Carbamimidoy...)
Affinity DataIC50:  3.10nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088978(CHEMBL176515 | N-[1-(1-Carbamimidoyl-2-hydroxy-pip...)
Affinity DataIC50:  5.10nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088984(2-Benzenesulfonylamino-N-[1-(1-carbamimidoyl-2-hyd...)
Affinity DataIC50:  10nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088979(CHEMBL366666 | {(R)-2-[2-((S)-1-Carbamimidoyl-2-hy...)
Affinity DataIC50:  11nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088985(CHEMBL369042 | {2-[2-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50:  12nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088977(CHEMBL177557 | {1-[1-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50:  19nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088987(CHEMBL174813 | {1-[1-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50:  23nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088986(CHEMBL433809 | {2-[2-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50:  101nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088985(CHEMBL369042 | {2-[2-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50:  125nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088981(CHEMBL425850 | {1-[1-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50:  261nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088978(CHEMBL176515 | N-[1-(1-Carbamimidoyl-2-hydroxy-pip...)
Affinity DataIC50:  275nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088982(CHEMBL160253 | CHEMBL367004 | N-[1-(1-Carbamimidoy...)
Affinity DataIC50:  367nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088979(CHEMBL366666 | {(R)-2-[2-((S)-1-Carbamimidoyl-2-hy...)
Affinity DataIC50:  482nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088981(CHEMBL425850 | {1-[1-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50:  699nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088977(CHEMBL177557 | {1-[1-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50:  904nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088984(2-Benzenesulfonylamino-N-[1-(1-carbamimidoyl-2-hyd...)
Affinity DataIC50:  1.17E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088987(CHEMBL174813 | {1-[1-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50:  1.46E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088983(CHEMBL177251 | {1-[1-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088984(2-Benzenesulfonylamino-N-[1-(1-carbamimidoyl-2-hyd...)
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088979(CHEMBL366666 | {(R)-2-[2-((S)-1-Carbamimidoyl-2-hy...)
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088987(CHEMBL174813 | {1-[1-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088983(CHEMBL177251 | {1-[1-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088980(CHEMBL177745 | {(R)-1-[(S)-1-((S)-1-Carbamimidoyl-...)
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088986(CHEMBL433809 | {2-[2-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088980(CHEMBL177745 | {(R)-1-[(S)-1-((S)-1-Carbamimidoyl-...)
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088985(CHEMBL369042 | {2-[2-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088983(CHEMBL177251 | {1-[1-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088982(CHEMBL160253 | CHEMBL367004 | N-[1-(1-Carbamimidoy...)
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088981(CHEMBL425850 | {1-[1-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088978(CHEMBL176515 | N-[1-(1-Carbamimidoyl-2-hydroxy-pip...)
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088977(CHEMBL177557 | {1-[1-(1-Carbamimidoyl-2-hydroxy-pi...)
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088980(CHEMBL177745 | {(R)-1-[(S)-1-((S)-1-Carbamimidoyl-...)
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed