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Found 14 Enz. Inhib. hit(s) with all data for entry = 50035193
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097337(CHEMBL349996 | Neamine derivative)
Affinity DataIC50:  28nMAssay Description:Inhibition of Tat peptide binding to HIV-1 TAR RNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Rev(Human immunodeficiency virus 1)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097337(CHEMBL349996 | Neamine derivative)
Affinity DataIC50:  350nMAssay Description:Compound was evaluated for its inhibitory activity against Klenow enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Rev(Human immunodeficiency virus 1)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097335(2-Amino-5-guanidino-pentanoic acid [(4R,5S,6S)-5-a...)
Affinity DataIC50:  460nMAssay Description:Inhibitory activity against peptide binding to the RRE RNA was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097335(2-Amino-5-guanidino-pentanoic acid [(4R,5S,6S)-5-a...)
Affinity DataIC50:  600nMAssay Description:Inhibition of Tat peptide binding to HIV-1 TAR RNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097336(CHEMBL152397 | Pyrene-1-carboxylic acid [(4R,5S,6S...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibitory concentration against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Rev(Human immunodeficiency virus 1)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097336(CHEMBL152397 | Pyrene-1-carboxylic acid [(4R,5S,6S...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibitory activity against peptide binding to the Rev Response Element RNA IIB was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Rev(Human immunodeficiency virus 1)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM8580((2R,3S,4R,5R,6R)-5-amino-2-(aminomethyl)-6-{[(1R,2...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibitory activity against peptide binding to the RRE RNA was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM8580((2R,3S,4R,5R,6R)-5-amino-2-(aminomethyl)-6-{[(1R,2...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of Tat peptide binding to HIV-1 TAR RNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Rev(Human immunodeficiency virus 1)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097337(CHEMBL349996 | Neamine derivative)
Affinity DataKd:  8.5nMAssay Description:Dissociation constant was determined for Rev Response Element RNA IIBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Rev(Human immunodeficiency virus 1)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097339(CHEMBL415806 | Neamine derivative)
Affinity DataKd:  3.40nMAssay Description:Dissociation constant was determined for Rev Response Element RNA IIBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097338(CHEMBL408877 | Neamine derivative)
Affinity DataKd:  25nMAssay Description:Dissociation constant for TAR RNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097337(CHEMBL349996 | Neamine derivative)
Affinity DataKd:  30nMAssay Description:Compound was evaluated for its inhibitory activity against Klenow enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Rev(Human immunodeficiency virus 1)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097336(CHEMBL152397 | Pyrene-1-carboxylic acid [(4R,5S,6S...)
Affinity DataKd:  240nMAssay Description:Inhibitory concentration against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097336(CHEMBL152397 | Pyrene-1-carboxylic acid [(4R,5S,6S...)
Affinity DataKd:  290nMAssay Description:Dissociation constant for TAR RNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed