Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50010773
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(CHEMBL266481 | GLUCAGON | His-Ser-Gln-Gly-Thr-Phe-...)
Affinity DataIC50:  1.5nMAssay Description:inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098563(CHEMBL413890 | Ser-Gln-Gly-Thr-Phe-Thr-Ser-Glu-Tyr...)
Affinity DataIC50:  3.75nMAssay Description:Compound was evaluated for its ability to displace radiolabelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098573(CHEMBL267876 | N-trinitrophenyl-His-Ser-Gln-Gly-Th...)
Affinity DataIC50:  15nMAssay Description:Compound was evaluated for its ability to displace radiolabelled glucagon (inactive up to 100 microM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098566(CHEMBL413208 | phenylbutyryl-Tyr-Ser-Lys-Tyr-Leu-A...)
Affinity DataIC50:  21.2nMAssay Description:IC50 value of the compound was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098572(Ac-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Tyr-Leu-Asp-Ser-Arg...)
Affinity DataIC50:  31nMAssay Description:IC50 value of the compound was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098570(CHEMBL438045 | Ser-Gln-Gly-Thr-Thr-Ser-Glu-Tyr-Ser...)
Affinity DataIC50:  48nMAssay Description:Compound was evaluated for its ability to displace radiolabelled glucagonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098565(Ac-Tyr-Ser-Lys-Tyr-Leu-Asp-Ser-Arg-Arg-Ala-Gln-Asp...)
Affinity DataIC50:  60nMAssay Description:IC50 value of the compound was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098567(CHEMBL439690 | phenylhexanoyl-Tyr-Ser-Lys-Tyr-Leu-...)
Affinity DataIC50:  131nMAssay Description:IC50 value of the compound was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098564(CHEMBL262418 | Phenacetyl-Tyr-Ser-Lys-Tyr-Leu-Asp-...)
Affinity DataIC50:  249nMAssay Description:IC50 value of the compound was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098574(CHEMBL409896 | phenylbutyryl-Tyr-Ser-Lys-2-Nal-Leu...)
Affinity DataIC50:  781nMAssay Description:IC50 value of the compound was expressed for inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098569(Ac-Nal-Ser-Lys-Nal-Leu-Asp-Ser-Arg-Arg-Ala-Gln-Asp...)
Affinity DataIC50:  800nMAssay Description:IC50 value of the compound was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Rattus norvegicus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50098568(Ac-Arg-Arg-Ala-Gln-Asp-Phe-Val-Gln-Trp-Leu-Met-Asn...)
Affinity DataIC50:  2.30E+3nMAssay Description:IC50 value of the compound was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed