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Found 30 Enz. Inhib. hit(s) with all data for entry = 50011427
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106478(CHEMBL443591 | FGGFTGARKCARKC)
Affinity DataIC50:  0.122nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106477(CHEMBL265801 | FGGFTGARKSARKLADE | Phe-GGFTGARKSAR...)
Affinity DataIC50:  0.286nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106479(CHEMBL384755 | FGGFTGARKSARK | H-FGGFTGARKSARK-NH2...)
Affinity DataIC50:  0.353nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106471(CHEMBL406718 | FGGFTGARKCARKC)
Affinity DataIC50:  0.471nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106480(CHEMBL437915 | FGGFTGARKSARKL)
Affinity DataIC50:  0.520nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106469(CHEMBL269029 | FGGFTCARKCARK | cyclo[Cys6,Cys10]N/...)
Affinity DataIC50:  0.833nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106470(CHEMBL442113 | FGGFTCARKCARK)
Affinity DataIC50:  3.03nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106476(CHEMBL435511 | FGGFTGCRKSCRK)
Affinity DataIC50:  3.04nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106468(CHEMBL424934 | FGGFTGCRKSARKC)
Affinity DataIC50:  4.97nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106475(CHEMBL266667 | FGGFTGCRKSCRK)
Affinity DataIC50:  8.70nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106467(CHEMBL384866 | FGGFTGCRKSARKC)
Affinity DataIC50:  37.2nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106481(CFGGFTGARKCARK | CHEMBL406010)
Affinity DataIC50:  387nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106472(CFGGFTCARKSARK | CHEMBL405451)
Affinity DataIC50:  874nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106474(CFGGFTGARKCARK | CHEMBL405948)
Affinity DataIC50:  1.29E+3nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106473(CFGGFTCARKSARK | CHEMBL268145)
Affinity DataIC50:  2.71E+3nMAssay Description:Displacement of [3H]-NC from human ORL1 receptor expressing HEK-293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106468(CHEMBL424934 | FGGFTGCRKSARKC)
Affinity DataEC50:  25nMAssay Description:Efficacy for human ORL1 receptor expressing HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106470(CHEMBL442113 | FGGFTCARKCARK)
Affinity DataEC50:  29.7nMAssay Description:Efficacy for human ORL1 receptor expressing HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106472(CFGGFTCARKSARK | CHEMBL405451)
Affinity DataEC50: >1.00E+4nMAssay Description:Efficacy for human ORL1 receptor expressing HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106481(CFGGFTGARKCARK | CHEMBL406010)
Affinity DataEC50:  439nMAssay Description:Efficacy for human ORL1 receptor expressing HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106477(CHEMBL265801 | FGGFTGARKSARKLADE | Phe-GGFTGARKSAR...)
Affinity DataEC50:  1.93nMAssay Description:Binding of compound to cell membranes expressing human ORL1 receptor in HEk-293 cells using [32S]-GTP-gammaSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106467(CHEMBL384866 | FGGFTGCRKSARKC)
Affinity DataEC50:  22.3nMAssay Description:Efficacy for human ORL1 receptor expressing HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106480(CHEMBL437915 | FGGFTGARKSARKL)
Affinity DataEC50:  1.97nMAssay Description:Efficacy for human ORL1 receptor expressing HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106473(CFGGFTCARKSARK | CHEMBL268145)
Affinity DataEC50: >1.00E+4nMAssay Description:Efficacy for human ORL1 receptor expressing HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106479(CHEMBL384755 | FGGFTGARKSARK | H-FGGFTGARKSARK-NH2...)
Affinity DataEC50:  1.12nMAssay Description:Efficacy for human ORL1 receptor expressing HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106471(CHEMBL406718 | FGGFTGARKCARKC)
Affinity DataEC50:  3.90nMAssay Description:Efficacy for human ORL1 receptor expressing HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106469(CHEMBL269029 | FGGFTCARKCARK | cyclo[Cys6,Cys10]N/...)
Affinity DataEC50:  31.3nMAssay Description:Efficacy for human ORL1 receptor expressing HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106478(CHEMBL443591 | FGGFTGARKCARKC)
Affinity DataEC50:  4.37nMAssay Description:Efficacy for human ORL1 receptor expressing HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106475(CHEMBL266667 | FGGFTGCRKSCRK)
Affinity DataEC50:  26.3nMAssay Description:Efficacy for human ORL1 receptor expressing HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106476(CHEMBL435511 | FGGFTGCRKSCRK)
Affinity DataEC50:  156nMAssay Description:Efficacy for human ORL1 receptor expressing HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106474(CFGGFTGARKCARK | CHEMBL405948)
Affinity DataEC50:  286nMAssay Description:Efficacy for human ORL1 receptor expressing HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed