Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50042224
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50115187(2-[2-carboxy-1-(3-methyl-1-(1-(2-Iodo-phenyl)-3-[4...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of Very late antigen 4 (VLA-4) and VCAM-Ig fusion protein interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50115186(3-(4-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetylamino}...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of Very late antigen 4 (VLA-4) and VCAM-Ig fusion protein interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50115176(2-Acetylamino-3-(4-{2-[4-(3-o-tolyl-ureido)-phenyl...)
Affinity DataIC50:  58nMAssay Description:Inhibition of Very late antigen 4 (VLA-4) and VCAM-Ig fusion protein interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50115177(CHEMBL103602 | [3-(3-{2-[4-(3-o-Tolyl-ureido)-phen...)
Affinity DataIC50:  67nMAssay Description:Inhibition of Very late antigen 4 (VLA-4) and VCAM-Ig fusion protein interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50115185(CHEMBL101126 | [(6-{2-[4-(3-o-Tolyl-ureido)-phenyl...)
Affinity DataIC50:  800nMAssay Description:Inhibition of Very late antigen 4 (VLA-4) and VCAM-Ig fusion protein interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50115182((3-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetylamino}-b...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Very late antigen 4 (VLA-4) and VCAM-Ig fusion protein interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50115181(3-Hydroxy-3-(3-{2-[4-(3-o-tolyl-ureido)-phenyl]-ac...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Very late antigen 4 (VLA-4) and VCAM-Ig fusion protein interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50115175((5-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetylamino}-[...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of Very late antigen 4 (VLA-4) and VCAM-Ig fusion protein interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50115180(3-(3-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetylamino}...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of Very late antigen 4 (VLA-4) and VCAM-Ig fusion protein interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50115183(3-(2-Methyl-4-{2-[4-(3-o-tolyl-ureido)-phenyl]-ace...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of Very late antigen 4 (VLA-4) and VCAM-Ig fusion protein interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50115179(3-(3-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetylamino}...)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of Very late antigen 4 (VLA-4) and VCAM-Ig fusion protein interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50115184((2-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetylamino}-t...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of Very late antigen 4 (VLA-4) and VCAM-Ig fusion protein interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50115178(3-(2-(1-Phenyl-vinyl)-3-{2-[4-(3-o-tolyl-ureido)-p...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of Very late antigen 4 (VLA-4) and VCAM-Ig fusion protein interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed