Compile Data Set for Download or QSAR
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Found 32 Enz. Inhib. hit(s) with all data for entry = 50013063
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125999((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  0.00205nMAssay Description:Ability of the compound to displace [3H]-DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126000((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataKi:  0.0216nMAssay Description:Ability of the compound to displace [3H]-DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126003((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataKi:  0.0350nMAssay Description:Ability of the compound to displace [3H]-DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125997((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataKi:  0.0618nMAssay Description:Ability of the compound to displace [3H]-DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125996((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataKi:  0.0623nMAssay Description:Ability of the compound to displace [3H]-DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125998((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataKi:  0.172nMAssay Description:Ability of the compound to displace [3H]-DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125999((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  1.10nMAssay Description:Ability of the compound to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126001((R)-2-((S)-2-Amino-3-phenyl-propionylamino)-5-guan...)
Affinity DataKi:  7.20nMAssay Description:Ability of the compound to displace [3H]-DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126002((R)-2-[(R)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataKi:  7.60nMAssay Description:Ability of the compound to displace [3H]-DAMGO from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125998((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataKi:  482nMAssay Description:Ability of the compound to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126003((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataKi:  544nMAssay Description:Ability of the compound to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126000((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataKi:  1.69E+3nMAssay Description:Ability of the compound to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125996((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataKi:  2.57E+3nMAssay Description:Ability of the compound to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125997((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataKi: >2.82E+3nMAssay Description:Ability of the compound to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126001((R)-2-((S)-2-Amino-3-phenyl-propionylamino)-5-guan...)
Affinity DataKi: >2.82E+3nMAssay Description:Ability of the compound to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126002((R)-2-[(R)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataKi: >2.82E+3nMAssay Description:Ability of the compound to displace [3H]-deltorphin II from delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125999((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataIC50:  0.0340nMAssay Description:Ability of the compound to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125999((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataIC50:  0.398nMAssay Description:Ability of the compound to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126003((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataIC50:  1.70nMAssay Description:Ability of the compound to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126000((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataIC50:  2.80nMAssay Description:Ability of the compound to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125998((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataIC50:  5.30nMAssay Description:Ability of the compound to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125996((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataIC50:  9.90nMAssay Description:Ability of the compound to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125997((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataIC50:  20nMAssay Description:Ability of the compound to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126003((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataIC50:  28nMAssay Description:Ability of the compound to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126000((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataIC50:  50nMAssay Description:Ability of the compound to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125998((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataIC50:  116nMAssay Description:Ability of the compound to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125996((R)-2-[(S)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataIC50:  188nMAssay Description:Ability of the compound to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50125997((R)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataIC50:  305nMAssay Description:Ability of the compound to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126002((R)-2-[(R)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataIC50:  320nMAssay Description:Ability of the compound to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126001((R)-2-((S)-2-Amino-3-phenyl-propionylamino)-5-guan...)
Affinity DataIC50:  633nMAssay Description:Ability of the compound to inhibit electrically induced contractions of guinea pig ileum having mu opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126002((R)-2-[(R)-2-Amino-3-(2,6-dimethyl-phenyl)-propion...)
Affinity DataIC50:  1.47E+3nMAssay Description:Ability of the compound to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Tohoku Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50126001((R)-2-((S)-2-Amino-3-phenyl-propionylamino)-5-guan...)
Affinity DataIC50:  7.14E+3nMAssay Description:Ability of the compound to inhibit electrically induced contractions of mouse vas deferens having delta opioid receptors tested in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed