Compile Data Set for Download or QSAR
maximum 50k data
Found 25 Enz. Inhib. hit(s) with all data for entry = 50000132
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001852(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-1-{2-[(3...)
Affinity DataIC50:  0.0450nMAssay Description:Binding ability towards opioid receptor mu expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001850((S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-[(...)
Affinity DataIC50:  0.130nMAssay Description:Binding ability towards opioid receptor mu expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001848(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-[1-met...)
Affinity DataIC50:  0.130nMAssay Description:Binding ability towards opioid receptor mu expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001846(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-[1-met...)
Affinity DataIC50:  0.5nMAssay Description:Binding ability towards opioid receptor mu expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001849(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-1-[2-(3-...)
Affinity DataIC50:  1.60nMAssay Description:Binding ability towards opioid receptor mu expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001845(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-[2-hyd...)
Affinity DataIC50:  1.70nMAssay Description:Binding ability towards opioid receptor mu expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001850((S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-[(...)
Affinity DataIC50:  4nMAssay Description:Binding ability towards opioid receptor delta expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001851(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-(1-met...)
Affinity DataIC50:  5.40nMAssay Description:Binding ability towards opioid receptor mu expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001853(2-Amino-N-(2-fluoro-1-methyl-6-phenyl-hex-2-enyl)-...)
Affinity DataIC50:  6.90nMAssay Description:Binding ability towards opioid receptor mu expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001852(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-1-{2-[(3...)
Affinity DataIC50:  10nMAssay Description:Binding ability towards opioid receptor kappa expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001852(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-1-{2-[(3...)
Affinity DataIC50:  12nMAssay Description:Binding ability towards opioid receptor delta expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001846(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-[1-met...)
Affinity DataIC50:  21nMAssay Description:Binding ability towards opioid receptor delta expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001847(2-Amino-N-[2-tert-butoxy-1-(3-phenyl-propoxymethyl...)
Affinity DataIC50:  33nMAssay Description:Binding ability towards opioid receptor mu expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001848(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-[1-met...)
Affinity DataIC50:  46nMAssay Description:Binding ability towards opioid receptor delta expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001849(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-1-[2-(3-...)
Affinity DataIC50:  110nMAssay Description:Binding ability towards opioid receptor delta expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001845(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-[2-hyd...)
Affinity DataIC50:  233nMAssay Description:Binding ability towards opioid receptor delta expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001849(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-1-[2-(3-...)
Affinity DataIC50:  280nMAssay Description:Binding ability towards opioid receptor kappa expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001848(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-[1-met...)
Affinity DataIC50:  330nMAssay Description:Binding ability towards opioid receptor kappa expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001847(2-Amino-N-[2-tert-butoxy-1-(3-phenyl-propoxymethyl...)
Affinity DataIC50:  340nMAssay Description:Binding ability towards opioid receptor delta expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001850((S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-[(...)
Affinity DataIC50:  380nMAssay Description:Binding ability towards opioid receptor kappa expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001846(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-[1-met...)
Affinity DataIC50:  1.30E+3nMAssay Description:Binding ability towards opioid receptor kappa expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001851(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-(1-met...)
Affinity DataIC50:  5.40E+3nMAssay Description:Binding ability towards opioid receptor kappa expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001845(2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-N-[2-hyd...)
Affinity DataIC50:  5.90E+3nMAssay Description:Binding ability towards opioid receptor kappa expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001853(2-Amino-N-(2-fluoro-1-methyl-6-phenyl-hex-2-enyl)-...)
Affinity DataIC50:  8.00E+3nMAssay Description:Binding ability towards opioid receptor kappa expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
G.D. Searle And

Curated by ChEMBL
LigandPNGBDBM50001847(2-Amino-N-[2-tert-butoxy-1-(3-phenyl-propoxymethyl...)
Affinity DataIC50:  9.30E+3nMAssay Description:Binding ability towards opioid receptor kappa expressed in homogenates of rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed