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Found 16 Enz. Inhib. hit(s) with all data for entry = 50036070
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50002313(2-Chloro-5-(2-{[2-(3-hydroxy-phenyl)-ethyl]-propyl...)
Affinity DataIC50:  730nMAssay Description:Inhibitory activity against [3H]spiperone in Rat Striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50002310(3-[2-(Phenethyl-propyl-amino)-ethyl]-phenol; hydro...)
Affinity DataIC50:  750nMAssay Description:Inhibitory activity against [3H]spiperone in Rat Striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50002314(2-Chloro-5-(2-{[3-(4-hydroxy-phenyl)-propyl]-propy...)
Affinity DataIC50:  850nMAssay Description:Inhibitory activity against [3H]spiperone in Rat Striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50002309(2-Chloro-5-(2-{[2-(4-hydroxy-phenyl)-ethyl]-propyl...)
Affinity DataIC50:  900nMAssay Description:Inhibitory activity against [3H]spiperone in Rat Striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50002311(2-Chloro-5-[2-(phenethyl-propyl-amino)-ethyl]-phen...)
Affinity DataIC50:  1.39E+3nMAssay Description:Inhibitory activity against [3H]spiperone in Rat Striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibitory activity against [3H]spiperone in Rat Striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibitory activity against [3H]-SCH- 23390 in Rat Striatal membraneMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50002313(2-Chloro-5-(2-{[2-(3-hydroxy-phenyl)-ethyl]-propyl...)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibitory activity against [3H]-SCH- 23390 in Rat Striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50002312(2-Chloro-5-(2-dipropylamino-ethyl)-phenol; hydrobr...)
Affinity DataIC50:  1.29E+4nMAssay Description:Inhibitory activity against [3H]spiperone in Rat Striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50002314(2-Chloro-5-(2-{[3-(4-hydroxy-phenyl)-propyl]-propy...)
Affinity DataIC50:  1.69E+4nMAssay Description:Inhibitory activity against [3H]-SCH- 23390 in Rat Striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50002309(2-Chloro-5-(2-{[2-(4-hydroxy-phenyl)-ethyl]-propyl...)
Affinity DataIC50:  1.81E+4nMAssay Description:Inhibitory activity against [3H]-SCH- 23390 in Rat Striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50002311(2-Chloro-5-[2-(phenethyl-propyl-amino)-ethyl]-phen...)
Affinity DataIC50:  2.44E+4nMAssay Description:Inhibitory activity against [3H]-SCH- 23390 in Rat Striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50002315(5-(2-Amino-ethyl)-2-chloro-phenol; hydrobromide | ...)
Affinity DataIC50:  2.53E+4nMAssay Description:Inhibitory activity against [3H]-SCH- 23390 in Rat Striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50002315(5-(2-Amino-ethyl)-2-chloro-phenol; hydrobromide | ...)
Affinity DataIC50:  2.63E+4nMAssay Description:Inhibitory activity against [3H]spiperone in Rat Striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50002312(2-Chloro-5-(2-dipropylamino-ethyl)-phenol; hydrobr...)
Affinity DataIC50:  5.07E+4nMAssay Description:Inhibitory activity against [3H]-SCH- 23390 in Rat Striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50002310(3-[2-(Phenethyl-propyl-amino)-ethyl]-phenol; hydro...)
Affinity DataIC50:  9.28E+4nMAssay Description:Inhibitory activity against [3H]-SCH- 23390 in Rat Striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed