Compile Data Set for Download or QSAR
maximum 50k data
Found 25 Enz. Inhib. hit(s) with all data for entry = 50000229
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003204(CHEMBL122438 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  0.0290nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003199(CHEMBL126008 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  0.0850nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003202(CHEMBL331408 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  0.480nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003200(CHEMBL267849 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  0.600nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003201(CHEMBL386376 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  0.910nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003196(CHEMBL433647 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003202(CHEMBL331408 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  2.10nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to Cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003201(CHEMBL386376 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  2.70nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding toCholecystokinin type A receptor in rat pancreatic membrane...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406690(CHEMBL2112635)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003200(CHEMBL267849 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003196(CHEMBL433647 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  4.90nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003207(CHEMBL405805 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  5nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003205(CHEMBL421471 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  9nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003203(CHEMBL436199 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  13nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003205(CHEMBL421471 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  22nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003204(CHEMBL122438 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  25nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to Cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003207(CHEMBL405805 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  73nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to Cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50406690(CHEMBL2112635)
Affinity DataIC50:  161nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to Cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50455666(CHEMBL2111823)
Affinity DataIC50:  165nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to Cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003203(CHEMBL436199 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  360nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003206(CHEMBL338056 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  1.20E+3nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003206(CHEMBL338056 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003199(CHEMBL126008 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  1.60E+3nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to Cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Bos taurus)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003198(CHEMBL124719 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of [3H]-propanoyl-CCK-8 binding to Cholecystokinin type B receptor in bovine striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50003198(CHEMBL124719 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50:  1.00E+4nMAssay Description:The compound was tested in vitro for inhibition of specific [3H]-propanoyl-CCK-8 binding to cholecystokinin type A receptor in rat pancreatic membran...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed