Affinity DataKi: 340nMAssay Description:Binding affinity determined by displacing [3H]DAMGO from Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Binding affinity determined by displacing [3H]DAMGO from Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 840nMAssay Description:Binding affinity determined by displacing [3H]DAMGO from Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.06E+3nMAssay Description:Binding affinity determined by displacing [3H][Ile5,6]deltorphin II from opioid receptor delta 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.84E+3nMAssay Description:Binding affinity determined by displacing [3H]U69,593 from Opioid receptor kappa 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.36E+3nMAssay Description:Binding affinity determined by displacing [3H]U69,593 from Opioid receptor kappa 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.06E+4nMAssay Description:Binding affinity determined by displacing [3H]DAMGO from Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.16E+4nMAssay Description:Binding affinity determined by displacing [3H]DAMGO from Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.38E+4nMAssay Description:Binding affinity determined by displacing [3H]DAMGO from Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.49E+4nMAssay Description:Binding affinity determined by displacing [3H]DAMGO from Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.69E+4nMAssay Description:Binding affinity determined by displacing [3H][Ile5,6]deltorphin II from opioid receptor delta 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.28E+4nMAssay Description:Binding affinity determined by displacing [3H]U69,593 from Opioid receptor kappa 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.79E+4nMAssay Description:Binding affinity determined by displacing [3H]DAMGO from Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.33E+4nMAssay Description:Binding affinity determined by displacing [3H]DAMGO from Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.49E+4nMAssay Description:Binding affinity determined by displacing [3H]DAMGO from Opioid receptor mu 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.62E+4nMAssay Description:Binding affinity determined by displacing [3H][Ile5,6]deltorphin II from opioid receptor delta 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.68E+4nMAssay Description:Binding affinity determined by displacing [3H]U69,593 from Opioid receptor kappa 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.09E+5nMAssay Description:Binding affinity determined by displacing [3H]U69,593 from Opioid receptor kappa 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+5nMAssay Description:Binding affinity determined by displacing [3H]U69,593 from Opioid receptor kappa 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.08E+5nMAssay Description:Binding affinity determined by displacing [3H]U69,593 from Opioid receptor kappa 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.13E+5nMAssay Description:Binding affinity determined by displacing [3H][Ile5,6]deltorphin II from opioid receptor delta 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.32E+5nMAssay Description:Binding affinity determined by displacing [3H][Ile5,6]deltorphin II from opioid receptor delta 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.61E+5nMAssay Description:Binding affinity determined by displacing [3H]U69,593 from Opioid receptor kappa 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.59E+5nMAssay Description:Binding affinity determined by displacing [3H]U69,593 from Opioid receptor kappa 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.14E+5nMAssay Description:Binding affinity determined by displacing [3H][Ile5,6]deltorphin II from opioid receptor delta 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.41E+5nMAssay Description:Binding affinity determined by displacing [3H]U69,593 from Opioid receptor kappa 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.65E+5nMAssay Description:Binding affinity determined by displacing [3H][Ile5,6]deltorphin II from opioid receptor delta 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 8.41E+5nMAssay Description:Binding affinity determined by displacing [3H][Ile5,6]deltorphin II from opioid receptor delta 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.17E+6nMAssay Description:Binding affinity determined by displacing [3H][Ile5,6]deltorphin II from opioid receptor delta 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.41E+6nMAssay Description:Binding affinity determined by displacing [3H][Ile5,6]deltorphin II from opioid receptor delta 1 in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 117nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human Opioid receptor kappa 1 ex...More data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human Opioid receptor mu 1 expre...More data for this Ligand-Target Pair
Affinity DataEC50: 9.80nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human Opioid receptor mu 1 expre...More data for this Ligand-Target Pair
Affinity DataEC50: 1.61E+3nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human opioid receptor delta 1 ex...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human Opioid receptor kappa 1 ex...More data for this Ligand-Target Pair
Affinity DataEC50: 87nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human opioid receptor delta 1 ex...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human Opioid receptor kappa 1 ex...More data for this Ligand-Target Pair
Affinity DataEC50: 21nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human opioid receptor delta 1 ex...More data for this Ligand-Target Pair
Affinity DataEC50: 4.5nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human Opioid receptor kappa 1 ex...More data for this Ligand-Target Pair
Affinity DataEC50: 7.90nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human opioid receptor delta 1 ex...More data for this Ligand-Target Pair
Affinity DataEC50: 1.11E+3nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human opioid receptor delta 1 ex...More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human Opioid receptor mu 1 expre...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human Opioid receptor mu 1 expre...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human Opioid receptor kappa 1 ex...More data for this Ligand-Target Pair
Affinity DataEC50: 3.5nMAssay Description:Concentration necessary to produce 50% of the Emax value, i.e. to stimulate [35S]GTP-gamma-S, binding to recombinant human Opioid receptor mu 1 expre...More data for this Ligand-Target Pair