Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 50000386
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005224(2-({Acetyl-[5-(16-methoxy-hexadecyloxy)-tetrahydro...)
Affinity DataIC50:  2.10nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005227(2-({Acetyl-[5-(6-decyloxy-hexyloxy)-tetrahydro-fur...)
Affinity DataIC50:  4.10nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005225(2-{[Acetyl-(5-hexadecyloxymethyl-tetrahydro-furan-...)
Affinity DataIC50:  8.60nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005231(2-{[Acetyl-(5-hexadecyloxy-tetrahydro-furan-3-ylme...)
Affinity DataIC50:  9.70nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005237(2-{[Acetyl-(5-octadecyloxymethyl-tetrahydro-furan-...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005232((R)-2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005229(2-{[Acetyl-(5-octadecyloxy-tetrahydro-furan-3-ylme...)
Affinity DataIC50:  13nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005230(2-[(Acetyl-{5-[6-(biphenyl-4-ylmethoxy)-hexyloxy]-...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005226(2-[(Acetyl-{5-[6-(5-phenyl-pentyloxy)-hexyloxy]-te...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005235(2-{[Acetyl-(5-octadecyloxy-tetrahydro-furan-3-ylme...)
Affinity DataIC50:  16nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005229(2-{[Acetyl-(5-octadecyloxy-tetrahydro-furan-3-ylme...)
Affinity DataIC50:  21nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005222(2-({Acetyl-[5-(6-oct-7-enyloxy-hexyloxy)-tetrahydr...)
Affinity DataIC50:  25nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005238(2-{[Acetyl-(5-octadecyloxy-tetrahydro-furan-3-ylme...)
Affinity DataIC50:  31nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005221(2-{[Acetyl-(5-icosyloxy-tetrahydro-furan-3-ylmetho...)
Affinity DataIC50:  40nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005228(2-[(Acetyl-{5-[6-(3-phenyl-propoxy)-hexyloxy]-tetr...)
Affinity DataIC50:  51nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005234(2-({Acetyl-[5-(3-phenyl-propoxy)-tetrahydro-furan-...)
Affinity DataIC50:  190nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005223(2-{[Acetyl-(5-heptadecyl-tetrahydro-furan-3-ylmeth...)
Affinity DataIC50:  210nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005233(2-({Acetyl-[5-(3,3-diphenyl-propoxy)-tetrahydro-fu...)
Affinity DataIC50:  260nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005240(2-({Acetyl-[5-(3-methyl-butoxy)-tetrahydro-furan-3...)
Affinity DataIC50:  690nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
J. Uriach & CíA.

Curated by ChEMBL
LigandPNGBDBM50005239(2-{[Acetyl-(5-ethoxy-tetrahydro-furan-3-ylmethoxyc...)
Affinity DataIC50:  2.80E+3nMAssay Description:In vitro inhibition of PAF induced aggregation of rabbit platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed