Compile Data Set for Download or QSAR
maximum 50k data
Found 59 Enz. Inhib. hit(s) with all data for entry = 50016529
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170132(1-Benzyl-7-methyl-3-propyl-1H,8H-imidazo[2,1-f]pur...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cells; range is 0.6 to 0.9 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170136(1-Benzyl-7-ethyl-3-propyl-1H,6H-pyrrolo[2,1-f]puri...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cells; range is 2.7 to 4.4 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170137(1-Benzyl-7-methyl-3-propyl-1H,6H-pyrrolo[2,1-f]pur...)
Affinity DataKi:  8nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170141(1-Benzyl-7-ethyl-3-propyl-1H,8H-imidazo[2,1-f]puri...)
Affinity DataKi:  15nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cells; range is 9 to 27More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170130(1-Benzyl-7-(4-fluoro-phenyl)-3-propyl-1H,8H-imidaz...)
Affinity DataKi:  22nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cells; range is 19 to 26 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170140(1-Benzyl-7-cyclopropyl-3-propyl-1H,8H-imidazo[2,1-...)
Affinity DataKi:  23nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cells; range is 18 to 29 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170139(1-Benzyl-7-isopropyl-3-propyl-1H,8H-imidazo[2,1-f]...)
Affinity DataKi:  31nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cells; range is 25 to 38More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170134(1-Benzyl-6,7-dimethyl-3-propyl-1H,8H-imidazo[2,1-f...)
Affinity DataKi:  36nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cells; range is 31 to 43 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170143(1-Benzyl-7-(4-methoxy-phenyl)-3-propyl-1H,8H-imida...)
Affinity DataKi:  55nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cells; range is 28 to 104 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170138(1-Benzyl-7-ethyl-6-methyl-3-propyl-1H,8H-imidazo[2...)
Affinity DataKi:  60nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cells; range is 53 to 69 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170142(1-Benzyl-6,7-dimethyl-3-propyl-1H,6H-pyrrolo[2,1-f...)
Affinity DataKi:  80nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170135(1-Benzyl-7-tert-butyl-3-propyl-1H,8H-imidazo[2,1-f...)
Affinity DataKi:  99nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cells; range is 77 to 129More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170128(1-Benzyl-7-phenyl-3-propyl-1H,8H-imidazo[2,1-f]pur...)
Affinity DataKi:  115nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170131(1-Benzyl-7-phenyl-3-propyl-1H,6H-pyrrolo[2,1-f]pur...)
Affinity DataKi:  200nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cells; range is 134 to 297 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170140(1-Benzyl-7-cyclopropyl-3-propyl-1H,8H-imidazo[2,1-...)
Affinity DataKi:  350nMAssay Description:Inhibition of [3H]-DPCPX binding to human A1 receptors expressed in CHO cells; range is 299 to 411More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170139(1-Benzyl-7-isopropyl-3-propyl-1H,8H-imidazo[2,1-f]...)
Affinity DataKi:  460nMAssay Description:Inhibition of [3H]-DPCPX binding to human A1 receptors expressed in CHO cells; range is 424 to 498More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170129(1-Benzyl-7-cyclohexyl-3-propyl-1H,8H-imidazo[2,1-f...)
Affinity DataKi:  555nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cells; range is 467 to 660 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170135(1-Benzyl-7-tert-butyl-3-propyl-1H,8H-imidazo[2,1-f...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170130(1-Benzyl-7-(4-fluoro-phenyl)-3-propyl-1H,8H-imidaz...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170128(1-Benzyl-7-phenyl-3-propyl-1H,8H-imidazo[2,1-f]pur...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170137(1-Benzyl-7-methyl-3-propyl-1H,6H-pyrrolo[2,1-f]pur...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170129(1-Benzyl-7-cyclohexyl-3-propyl-1H,8H-imidazo[2,1-f...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170133(1-Benzyl-7-biphenyl-4-yl-3-propyl-1H,8H-imidazo[2,...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170131(1-Benzyl-7-phenyl-3-propyl-1H,6H-pyrrolo[2,1-f]pur...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170137(1-Benzyl-7-methyl-3-propyl-1H,6H-pyrrolo[2,1-f]pur...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170131(1-Benzyl-7-phenyl-3-propyl-1H,6H-pyrrolo[2,1-f]pur...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170134(1-Benzyl-6,7-dimethyl-3-propyl-1H,8H-imidazo[2,1-f...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170129(1-Benzyl-7-cyclohexyl-3-propyl-1H,8H-imidazo[2,1-f...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170133(1-Benzyl-7-biphenyl-4-yl-3-propyl-1H,8H-imidazo[2,...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170132(1-Benzyl-7-methyl-3-propyl-1H,8H-imidazo[2,1-f]pur...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170140(1-Benzyl-7-cyclopropyl-3-propyl-1H,8H-imidazo[2,1-...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170143(1-Benzyl-7-(4-methoxy-phenyl)-3-propyl-1H,8H-imida...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170138(1-Benzyl-7-ethyl-6-methyl-3-propyl-1H,8H-imidazo[2...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170134(1-Benzyl-6,7-dimethyl-3-propyl-1H,8H-imidazo[2,1-f...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170143(1-Benzyl-7-(4-methoxy-phenyl)-3-propyl-1H,8H-imida...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170139(1-Benzyl-7-isopropyl-3-propyl-1H,8H-imidazo[2,1-f]...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170133(1-Benzyl-7-biphenyl-4-yl-3-propyl-1H,8H-imidazo[2,...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170138(1-Benzyl-7-ethyl-6-methyl-3-propyl-1H,8H-imidazo[2...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170130(1-Benzyl-7-(4-fluoro-phenyl)-3-propyl-1H,8H-imidaz...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170128(1-Benzyl-7-phenyl-3-propyl-1H,8H-imidazo[2,1-f]pur...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170141(1-Benzyl-7-ethyl-3-propyl-1H,8H-imidazo[2,1-f]puri...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170142(1-Benzyl-6,7-dimethyl-3-propyl-1H,6H-pyrrolo[2,1-f...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170141(1-Benzyl-7-ethyl-3-propyl-1H,8H-imidazo[2,1-f]puri...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170142(1-Benzyl-6,7-dimethyl-3-propyl-1H,6H-pyrrolo[2,1-f...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170136(1-Benzyl-7-ethyl-3-propyl-1H,6H-pyrrolo[2,1-f]puri...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170136(1-Benzyl-7-ethyl-3-propyl-1H,6H-pyrrolo[2,1-f]puri...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170132(1-Benzyl-7-methyl-3-propyl-1H,8H-imidazo[2,1-f]pur...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170135(1-Benzyl-7-tert-butyl-3-propyl-1H,8H-imidazo[2,1-f...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM 241385 binding to human adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170137(1-Benzyl-7-methyl-3-propyl-1H,6H-pyrrolo[2,1-f]pur...)
Affinity DataIC50:  400nMAssay Description:Inhibition of 100 nM NECA-stimulated cAMP production in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170138(1-Benzyl-7-ethyl-6-methyl-3-propyl-1H,8H-imidazo[2...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of 100 nM NECA-stimulated cAMP production in CHO cells expressing human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 59 total ) | Next | Last >>
Jump to: