Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 50024708
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(CHEMBL499519 | GNF-PF-5618 | nocardimicin B)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(CHEMBL499519 | GNF-PF-5618 | nocardimicin B)
Affinity DataKi:  140nMAssay Description:Binding affinity to human muscarinic M4 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241915(CHEMBL450986 | nocardimicin D)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(CHEMBL499519 | GNF-PF-5618 | nocardimicin B)
Affinity DataKi:  490nMAssay Description:Binding affinity to human muscarinic M1 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(CHEMBL499519 | GNF-PF-5618 | nocardimicin B)
Affinity DataKi:  630nMAssay Description:Binding affinity to human muscarinic M2 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241916(CHEMBL510340 | Noccardimicin E)
Affinity DataKi:  970nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241914(CHEMBL507760 | nocardimicin C)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(CHEMBL499519 | GNF-PF-5618 | nocardimicin B)
Affinity DataKi:  1.18E+3nMAssay Description:Binding affinity to human muscarinic M5 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241912(CHEMBL505197 | Nocardimicin A)
Affinity DataKi:  1.25E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241917(CHEMBL508807 | Nocardimicin F)
Affinity DataKi:  1.33E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(CHEMBL499519 | GNF-PF-5618 | nocardimicin B)
Affinity DataIC50:  630nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(CHEMBL499519 | GNF-PF-5618 | nocardimicin B)
Affinity DataIC50:  1.04E+3nMAssay Description:Binding affinity to human muscarinic M4 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241915(CHEMBL450986 | nocardimicin D)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(CHEMBL499519 | GNF-PF-5618 | nocardimicin B)
Affinity DataIC50:  1.64E+3nMAssay Description:Binding affinity to human muscarinic M5 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(CHEMBL499519 | GNF-PF-5618 | nocardimicin B)
Affinity DataIC50:  1.78E+3nMAssay Description:Binding affinity to human muscarinic M2 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241913(CHEMBL499519 | GNF-PF-5618 | nocardimicin B)
Affinity DataIC50:  2.03E+3nMAssay Description:Binding affinity to human muscarinic M1 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241916(CHEMBL510340 | Noccardimicin E)
Affinity DataIC50:  4.56E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241914(CHEMBL507760 | nocardimicin C)
Affinity DataIC50:  4.70E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241912(CHEMBL505197 | Nocardimicin A)
Affinity DataIC50:  5.89E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50241917(CHEMBL508807 | Nocardimicin F)
Affinity DataIC50:  6.29E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed