Compile Data Set for Download or QSAR
maximum 50k data
Found 50 Enz. Inhib. hit(s) with all data for entry = 50016772
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173419((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-{(E)-2-[5-(3-tr...)
Affinity DataKi:  2.70nMAssay Description:Inhibitory constant aganist Protease-activated receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173417((3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-ethylpyridin-2-yl)...)
Affinity DataKi:  12nMAssay Description:Inhibitory constant aganist Protease-activated receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173437((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(3-Chloro-phen...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173419((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-{(E)-2-[5-(3-tr...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173433((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(2-Methoxy-phe...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173419((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-{(E)-2-[5-(3-tr...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173409((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(5-m-tol...)
Affinity DataIC50:  13nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173410((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(5-o-tol...)
Affinity DataIC50:  14nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173418((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(3-Isopropyl-p...)
Affinity DataIC50:  19nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173451((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(5-Benzyloxy-pyri...)
Affinity DataIC50:  19nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173417((3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-ethylpyridin-2-yl)...)
Affinity DataIC50:  20nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173438((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(2-Fluoro-phen...)
Affinity DataIC50:  22nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173436(3-{6-[(E)-2-((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-1-ox...)
Affinity DataIC50:  25nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173430((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(3-Bromo-pheny...)
Affinity DataIC50:  25nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173447((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(2-Chloro-phen...)
Affinity DataIC50:  26nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173421((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(5-pheny...)
Affinity DataIC50:  27nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173446((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(3-Methoxy-phe...)
Affinity DataIC50:  28nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173445((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(3-Fluoro-phen...)
Affinity DataIC50:  35nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173419((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-{(E)-2-[5-(3-tr...)
Affinity DataIC50:  44nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173434(2-{6-[(E)-2-((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-1-ox...)
Affinity DataIC50:  44nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173450((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-{(E)-2-[5-(2-tr...)
Affinity DataIC50:  46nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173417((3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-ethylpyridin-2-yl)...)
Affinity DataIC50:  85nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173417((3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-ethylpyridin-2-yl)...)
Affinity DataIC50:  85nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173431(3-{6-[(E)-2-((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-1-ox...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173415((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Butyl-pyridin-...)
Affinity DataIC50:  143nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173424((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(6-vinyl...)
Affinity DataIC50:  150nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173426((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(4-Methoxy-phe...)
Affinity DataIC50:  204nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173427((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Cyclopropyl-py...)
Affinity DataIC50:  210nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173449((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(6-propy...)
Affinity DataIC50:  250nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173425((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(6-methy...)
Affinity DataIC50:  300nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173425((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(6-methy...)
Affinity DataIC50:  300nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173412((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-{(E)-2-[5-(4-tr...)
Affinity DataIC50: >300nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173414((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(5-Methoxy-pyridi...)
Affinity DataIC50:  325nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173420((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(5-p-tol...)
Affinity DataIC50:  325nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173411((3S,3aR,4R,4aS,8aR,9aS)-4-[(E)-2-(6-Ethyl-pyridin-...)
Affinity DataIC50:  400nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173443((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(4-Fluoro-phen...)
Affinity DataIC50:  467nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173422((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Isobutyl-pyrid...)
Affinity DataIC50:  550nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173439((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Isopropyl-pyri...)
Affinity DataIC50:  725nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173440((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Methoxymethyl-...)
Affinity DataIC50:  850nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173444((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Benzyl-pyridin...)
Affinity DataIC50:  900nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173432((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(4-Chloro-phen...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173429((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(5-methy...)
Affinity DataIC50:  1.10E+3nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173441((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(6-methy...)
Affinity DataIC50:  1.25E+3nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173442((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[(E)-2-(6-methy...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173428((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Hydroxymethyl-...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173413((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(4-methy...)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173435((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Hexyl-pyridin-...)
Affinity DataIC50:  3.50E+3nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173448((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(5-Benzyl-pyridin...)
Affinity DataIC50:  3.68E+3nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173416((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-((E)-2-pyridin-...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50173423((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(3-methy...)
Affinity DataIC50: >5.00E+3nMAssay Description:In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed