Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50017143
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Umr Cnrs/Ulp 7081

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  23.5nMAssay Description:Displacement of [3H]QNB from EGFP(delta17)human M1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Umr Cnrs/Ulp 7081

Curated by ChEMBL
LigandPNGBDBM50178133(1-ethyl-2-[(1E,3E)-3-(1-ethylquinolin-2-(1H)-ylide...)
Affinity DataKi:  29.4nMAssay Description:Displacement of [3H]QNB from EGFP(delta17)human M1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Umr Cnrs/Ulp 7081

Curated by ChEMBL
LigandPNGBDBM50178130(CHEMBL220095 | RR(17)PZ)
Affinity DataKi:  53.5nMAssay Description:Displacement of [3H]QNB from EGFP(delta17)human M1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Umr Cnrs/Ulp 7081

Curated by ChEMBL
LigandPNGBDBM50178128(Bo(15)PZ | CHEMBL198982)
Affinity DataKi:  69.7nMAssay Description:Displacement of [3H]QNB from EGFP(delta17)human M1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Umr Cnrs/Ulp 7081

Curated by ChEMBL
LigandPNGBDBM50178129(2-{[4-(diethylamino)phenyl][4-(diethyliminio)cyclo...)
Affinity DataKi:  189nMAssay Description:Displacement of [3H]QNB from EGFP(delta17)human M1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Umr Cnrs/Ulp 7081

Curated by ChEMBL
LigandPNGBDBM50178132(CHEMBL370564 | {4-[[4-(5-carboxy-pentylsulfamoyl)-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]QNB from EGFP(delta17)human M1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Umr Cnrs/Ulp 7081

Curated by ChEMBL
LigandPNGBDBM50178131(6-[(5-carboxypentanoyl)amino]-1-ethyl-2-[(1E,3E)-3...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]QNB from EGFP(delta17)human M1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed