Compile Data Set for Download or QSAR
maximum 50k data
Found 26 Enz. Inhib. hit(s) with all data for entry = 50017271
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50063882((6aR,10aR)-3-(hept-1-ynyl)-6,6,9-trimethyl-6a,7,10...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [3H]CP-55,940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50063882((6aR,10aR)-3-(hept-1-ynyl)-6,6,9-trimethyl-6a,7,10...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]CP-55,940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179985(1-((6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10...)
Affinity DataKi:  3.86nMAssay Description:Displacement of [3H]CP-55,940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50169951((6aR,10aR)-3-Adamantan-1-yl-6,6,9-trimethyl-6a,7,1...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]CP-55,940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179985(1-((6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10...)
Affinity DataKi:  8.26nMAssay Description:Displacement of [3H]CP-55,940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179978((6aR,10aR)-6,6,9-trimethyl-3-(naphthalen-1-yl)-6a,...)
Affinity DataKi:  9.39nMAssay Description:Displacement of [3H]CP-55,940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179978((6aR,10aR)-6,6,9-trimethyl-3-(naphthalen-1-yl)-6a,...)
Affinity DataKi:  11.7nMAssay Description:Displacement of [3H]CP-55,940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179980(1-((6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10...)
Affinity DataKi:  25.2nMAssay Description:Displacement of [3H]CP-55,940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179980(1-((6aR,10aR)-1-hydroxy-6,6,9-trimethyl-6a,7,10,10...)
Affinity DataKi:  27.9nMAssay Description:Displacement of [3H]CP-55,940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50067734((-)-(6aR-trans)-6,6,9-trimethyl-3-pentyl-6a,7,10,1...)
Affinity DataKi:  39.3nMAssay Description:Displacement of [3H]CP-55,940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50067734((-)-(6aR-trans)-6,6,9-trimethyl-3-pentyl-6a,7,10,1...)
Affinity DataKi:  47.6nMAssay Description:Displacement of [3H]CP-55,940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179986((6aR,10aR)-3-(4-ethyl-phenyl)-6,6,9-trimethyl-6a,7...)
Affinity DataKi:  51.7nMAssay Description:Displacement of [3H]CP-55,940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50169951((6aR,10aR)-3-Adamantan-1-yl-6,6,9-trimethyl-6a,7,1...)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]CP-55,940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179983((6aR,10aR)-6,6,9-trimethyl-3-(4-propyl-phenyl)-6a,...)
Affinity DataKi:  57.8nMAssay Description:Displacement of [3H]CP-55,940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179982((6aR,10aR)-6,6,9-trimethyl-3-p-tolyl-6a,7,10,10a-t...)
Affinity DataKi:  71.8nMAssay Description:Displacement of [3H]CP-55,940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179982((6aR,10aR)-6,6,9-trimethyl-3-p-tolyl-6a,7,10,10a-t...)
Affinity DataKi:  95.5nMAssay Description:Displacement of [3H]CP-55,940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179981(1-[3,5-dihydroxy-4-((1R,6R)-6-isopropenyl-3-methyl...)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]CP-55,940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179983((6aR,10aR)-6,6,9-trimethyl-3-(4-propyl-phenyl)-6a,...)
Affinity DataKi:  108nMAssay Description:Displacement of [3H]CP-55,940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179987(1-[3,5-dihydroxy-4-((1R,6R)-6-isopropenyl-3-methyl...)
Affinity DataKi:  111nMAssay Description:Displacement of [3H]CP-55,940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179986((6aR,10aR)-3-(4-ethyl-phenyl)-6,6,9-trimethyl-6a,7...)
Affinity DataKi:  119nMAssay Description:Displacement of [3H]CP-55,940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179984(2-((1R,6R)-6-isopropenyl-3-methyl-cyclohex-2-enyl)...)
Affinity DataKi:  222nMAssay Description:Displacement of [3H]CP-55,940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179981(1-[3,5-dihydroxy-4-((1R,6R)-6-isopropenyl-3-methyl...)
Affinity DataKi:  255nMAssay Description:Displacement of [3H]CP-55,940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179987(1-[3,5-dihydroxy-4-((1R,6R)-6-isopropenyl-3-methyl...)
Affinity DataKi:  319nMAssay Description:Displacement of [3H]CP-55,940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(MOUSE)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179979(4-((1R,6R)-6-isopropenyl-3-methyl-cyclohex-2-enyl)...)
Affinity DataKi:  374nMAssay Description:Displacement of [3H]CP-55,940 from mouse spleen CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179979(4-((1R,6R)-6-isopropenyl-3-methyl-cyclohex-2-enyl)...)
Affinity DataKi:  638nMAssay Description:Displacement of [3H]CP-55,940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50179984(2-((1R,6R)-6-isopropenyl-3-methyl-cyclohex-2-enyl)...)
Affinity DataKi:  754nMAssay Description:Displacement of [3H]CP-55,940 from rat brain CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed